Discovery of 4-oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate (ML221) as a functional antagonist of the apelin (APJ) receptor
发现 4-氧代-6-((嘧啶-2-基硫代)甲基)-4H-吡喃-3-基 4-硝基苯甲酸酯 (ML221) 是阿扑素 (APJ) 受体的功能性拮抗剂
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.5
doi:10.1016/j.bmcl.2012.08.105
Patrick R Maloney, Pasha Khan, Michael Hedrick, Palak Gosalia, Monika Milewski, Linda Li, Gregory P Roth, Eduard Sergienko, Eigo Suyama, Eliot Sugarman, Kevin Nguyen, Alka Mehta, Stefan Vasile, Ying Su, Derek Stonich, Hung Nguyen, Fu-Yue Zeng, Arianna Mangravita Novo, Michael Vicchiarelli, Jena Diwa