日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MondoA coordinately regulates skeletal myocyte lipid homeostasis and insulin signaling

MondoA 协调调节骨骼肌细胞脂质稳态和胰岛素信号

Byungyong Ahn, Mangala M Soundarapandian, Hampton Sessions, Satyamaheshwar Peddibhotla, Gregory P Roth, Jian-Liang Li, Eliot Sugarman, Ada Koo, Siobhan Malany, Miao Wang, Kyungmoo Yea, Jeanne Brooks, Teresa C Leone, Xianlin Han, Rick B Vega, Daniel P Kelly

Nrf2 and HSF-1 Pathway Activation via Hydroquinone-Based Proelectrophilic Small Molecules is Regulated by Electrochemical Oxidation Potential

基于氢醌的亲电小分子激活Nrf2和HSF-1通路受电化学氧化电位调控

Takumi Satoh ,Romain Stalder ,Scott R McKercher ,Robert E Williamson ,Gregory P Roth ,Stuart A Lipton

Imidazole-derived agonists for the neurotensin 1 receptor

咪唑衍生物的神经降压素 1 受体激动剂

Paul M Hershberger, Michael P Hedrick, Satyamaheshwar Peddibhotla, Arianna Mangravita-Novo, Palak Gosalia, Yujie Li, Wilson Gray, Michael Vicchiarelli, Layton H Smith, Thomas D Y Chung, James B Thomas, Marc G Caron, Anthony B Pinkerton, Lawrence S Barak, Gregory P Roth

Discovery of 4-oxo-6-((pyrimidin-2-ylthio)methyl)-4H-pyran-3-yl 4-nitrobenzoate (ML221) as a functional antagonist of the apelin (APJ) receptor

发现 4-氧代-6-((嘧啶-2-基硫代)甲基)-4H-吡喃-3-基 4-硝基苯甲酸酯 (ML221) 是阿扑素 (APJ) 受体的功能性拮抗剂

Patrick R Maloney, Pasha Khan, Michael Hedrick, Palak Gosalia, Monika Milewski, Linda Li, Gregory P Roth, Eduard Sergienko, Eigo Suyama, Eliot Sugarman, Kevin Nguyen, Alka Mehta, Stefan Vasile, Ying Su, Derek Stonich, Hung Nguyen, Fu-Yue Zeng, Arianna Mangravita Novo, Michael Vicchiarelli, Jena Diwa

Dual neuroprotective pathways of a pro-electrophilic compound via HSF-1-activated heat-shock proteins and Nrf2-activated phase 2 antioxidant response enzymes

促电化合物通过 HSF-1 激活的热休克蛋白和 Nrf2 激活的 2 期抗氧化反应酶发挥双重神经保护作用

Takumi Satoh ,Tayebeh Rezaie, Masaaki Seki, Carmen R Sunico, Takahito Tabuchi, Tomomi Kitagawa, Mika Yanagitai, Mutsumi Senzaki, Chihiro Kosegawa, Hideharu Taira, Scott R McKercher, Jennifer K Hoffman, Gregory P Roth, Stuart A Lipton

Chemical genetics approach to restoring p27Kip1 reveals novel compounds with antiproliferative activity in prostate cancer cells

恢复 p27Kip1 的化学遗传学方法揭示了在前列腺癌细胞中具有抗增殖活性的新型化合物

Elizabeth Rico-Bautista, Chih-Cheng Yang, Lifang Lu, Gregory P Roth, Dieter A Wolf