日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mitochondrial KMT9 methylates DLAT to control pyruvate dehydrogenase activity and prostate cancer growth

线粒体KMT9通过甲基化DLAT来控制丙酮酸脱氢酶活性和前列腺癌生长。

Jia, Yanhan; Wang, Sheng; Urban, Sylvia; Müller, Judith M; Sum, Manuela; Wang, Qing; Bauer, Helena; Schulte, Uwe; Rampelt, Heike; Pfanner, Nikolaus; Schüle, Katrin M; Imhof, Axel; Forné, Ignasi; Berlin, Christopher; Sigle, August; Gratzke, Christian; Greschik, Holger; Metzger, Eric; Schüle, Roland

Molecular determinants for recognition of serotonylated chromatin

识别血清素化染色质的分子决定因素

Pulido-Cortés, Laura; Gielingh, Hajo; Thijssen, Vito; Liu, Minglong; Yoshisada, Ryoji; Romão Soares, Leonardo; Nizamuddin, Sheikh; Friedrich, Florian; Greschik, Holger; Peng, Ling; Vargas Honorato, Rodrigo; Jung, Manfred; Bonvin, Alexandre M J J; Biniossek, Martin L; Schüle, Roland; Jongkees, Seino; van Ingen, Hugo; Timmers, H Th Marc

Structure-guided design of a selective inhibitor of the methyltransferase KMT9 with cellular activity

具有细胞活性的甲基转移酶 KMT9 选择性抑制剂的结构引导设计

Sheng Wang, Sebastian O Klein, Sylvia Urban, Maximilian Staudt, Nicolas P F Barthes, Dominica Willmann, Johannes Bacher, Manuela Sum, Helena Bauer, Ling Peng, Georg A Rennar, Christian Gratzke, Katrin M Schüle, Lin Zhang, Oliver Einsle, Holger Greschik, Calum MacLeod, Christopher G Thomson, Manfred

Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor

发现一种高效、选择性强且具有细胞活性的SPIN1抑制剂

Xiong, Yan; Greschik, Holger; Johansson, Catrine; Seifert, Ludwig; Gamble, Vicki; Park, Kwang-Su; Fagan, Vincent; Li, Fengling; Chau, Irene; Vedadi, Masoud; Arrowsmith, Cheryl H; Brennan, Paul; Fedorov, Oleg; Jung, Manfred; Farnie, Gillian; Liu, Jing; Oppermann, Udo; Schüle, Roland; Jin, Jian

Lysine Methyltransferase 9 (KMT9) Is an Actionable Target in Muscle-Invasive Bladder Cancer

赖氨酸甲基转移酶 9 (KMT9) 是肌肉浸润性膀胱癌的可行靶点

Sainab Totonji, Anna Ramos-Triguero, Dominica Willmann, Manuela Sum, Sylvia Urban, Helena Bauer, Astrid Rieder, Sheng Wang, Holger Greschik, Eric Metzger, Roland Schüle

Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors

基于结构的A366衍生物作为Spindlin1抑制剂的设计、对接和结合自由能计算

Luise, Chiara; Robaa, Dina; Regenass, Pierre; Maurer, David; Ostrovskyi, Dmytro; Seifert, Ludwig; Bacher, Johannes; Burgahn, Teresa; Wagner, Tobias; Seitz, Johannes; Greschik, Holger; Park, Kwang-Su; Xiong, Yan; Jin, Jian; Schüle, Roland; Breit, Bernhard; Jung, Manfred; Sippl, Wolfgang

The histone code reader Spin1 controls skeletal muscle development

组蛋白密码阅读器 Spin1 控制骨骼肌发育

Holger Greschik, Delphine Duteil, Nadia Messaddeq, Dominica Willmann, Laura Arrigoni, Manuela Sum, Manfred Jung, Daniel Metzger, Thomas Manke, Thomas Günther, Roland Schüle

Chronic non-bacterial osteitis from the patient perspective: a health services research through data collected from patient conferences

从患者角度看慢性非细菌性骨炎:一项基于患者会议数据的健康服务研究

Silier, Colen Cooper Gore; Greschik, Justina; Gesell, Susanne; Grote, Veit; Jansson, Annette F

Identification of a small-molecule ligand of the epigenetic reader protein Spindlin1 via a versatile screening platform

通过多功能筛选平台鉴定表观遗传读取蛋白 Spindlin1 的小分子配体

Tobias Wagner, Holger Greschik, Teresa Burgahn, Karin Schmidtkunz, Anne-Kathrin Schott, Joel McMillan, Lina Baranauskienė, Yan Xiong, Oleg Fedorov, Jian Jin, Udo Oppermann, Daumantas Matulis, Roland Schüle, Manfred Jung

The histone code reader SPIN1 controls RET signaling in liposarcoma

组蛋白密码阅读器 SPIN1 控制脂肪肉瘤中的 RET 信号传导

Henriette Franz, Holger Greschik, Dominica Willmann, Luka Ozretić, Cordula Annette Jilg, Eva Wardelmann, Manfred Jung, Reinhard Buettner, Roland Schüle