Axitinib effectively inhibits BCR-ABL1(T315I) with a distinct binding conformation
阿昔替尼通过独特的结合构象有效抑制 BCR-ABL1(T315I)
期刊:Nature
影响因子:50.5
doi:10.1038/nature14119
Tea Pemovska, Eric Johnson, Mika Kontro, Gretchen A Repasky, Jeffrey Chen, Peter Wells, Ciarán N Cronin, Michele McTigue, Olli Kallioniemi, Kimmo Porkka, Brion W Murray, Krister Wennerberg