日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Experimental and machine learning-based exploration of repurposed drugs reveals chemical features underlying phospholipidosis

通过实验和机器学习方法对现有药物进行探索,揭示了磷脂沉积症的潜在化学特征。

Kuzikov, Maria; Kalman, Adelinn; Karki, Reagon; Reinshagen, Jeanette; Huchting, Johanna; Qian, Kun; Axelsson, Hanna; Tampere, Marianna; Östling, Päivi; Seashore-Ludlow, Brinton; Gadiya, Yojana; Gribbon, Philip; Zaliani, Andrea

The COMBINE pneumonia model: a multicenter study to standardize a mouse pneumonia model with Pseudomonas aeruginosa and Klebsiella pneumoniae for antibiotic development

COMBINE肺炎模型:一项多中心研究,旨在标准化铜绿假单胞菌和肺炎克雷伯菌小鼠肺炎模型,用于抗生素研发

Hansen, Jon U; Arrazuria, Rakel; Hoover, Jennifer L; Kerscher, Bernhard; Huseby, Douglas L; Sordello, Sylvie; Gribbon, Philip; Gadiya, Yojana; Berlin, Leonie von; Witt, Gesa; Tassi, Natália; Rosenborg, Frederikke; Cao, Sha; Bekeredjian-Ding, Isabelle; Lindahl, Otto; Hughes, Diarmaid; Friberg, Lena E; Vingsbo Lundberg, Carina

ECBD: European chemical biology database

ECBD:欧洲化学生物学数据库

Škuta, Ctibor; Müller, Tomáš; Voršilák, Milan; Popr, Martin; Epp, Trevor; Skopelitou, Katholiki E; Rossella, Federica; Stechmann, Bahne; Gribbon, Philip; Bartůněk, Petr

Lessons Learned From European Health Data Projects With Cancer Use Cases: Implementation of Health Standards and Internet of Things Semantic Interoperability

从欧洲健康数据项目中汲取的癌症应用案例经验教训:健康标准和物联网语义互操作性的实施

Gyrard, Amelie; Abedian, Somayeh; Gribbon, Philip; Manias, George; van Nuland, Rick; Zatloukal, Kurt; Nicolae, Irina Emilia; Danciu, Gabriel; Nechifor, Septimiu; Marti-Bonmati, Luis; Mallol, Pedro; Dalmiani, Stefano; Autexier, Serge; Jendrossek, Mario; Avramidis, Ioannis; Garcia Alvarez, Eva; Holub, Petr; Blanquer, Ignacio; Boden, Anna; Hussein, Rada

Interoperability Framework of the European Health Data Space for the Secondary Use of Data: Interactive European Interoperability Framework-Based Standards Compliance Toolkit for AI-Driven Projects

欧洲健康数据空间数据二次利用互操作性框架:面向人工智能驱动项目的交互式欧洲互操作性框架标准合规性工具包

Hussein, Rada; Gyrard, Amelie; Abedian, Somayeh; Gribbon, Philip; Martínez, Sara Alabart

Predicting Antimicrobial Class Specificity of Small Molecules Using Machine Learning

利用机器学习预测小分子抗菌药物的类别特异性

Gadiya, Yojana; Genilloud, Olga; Bilitewski, Ursula; Brönstrup, Mark; von Berlin, Leonie; Attwood, Marie; Gribbon, Philip; Zaliani, Andrea

Papaverine Targets STAT Signaling: A Dual-Action Therapy Option Against SARS-CoV-2.

罂粟碱靶向 STAT 信号通路:对抗 SARS-CoV-2 的双重作用疗法选择

Reus Philipp, Torbica Emma, Rothenburger Tamara, Bechtel Marco, Kandler Joshua, Ciesek Sandra, Gribbon Philip, Kannt Aimo, Cinatl Jindrich, Bojkova Denisa

Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2.

硫醇反应性或氧化还原活性:修改重新定位筛选导致新的无效化流程,并鉴定出针对 SARS-CoV-2 木瓜蛋白酶样蛋白酶的真正非共价抑制剂

Kuzikov Maria, Morasso Stefano, Reinshagen Jeanette, Wolf Markus, Monaco Vittoria, Cozzolino Flora, Golič Grdadolnik Simona, Šket Primož, Plavec Janez, Iaconis Daniela, Summa Vincenzo, Corona Angela, Paulis Annalaura, Esposito Francesca, Tramontano Enzo, Monti Maria, Beccari Andrea R, Manelfi Candida, Windshügel Björn, Gribbon Philip, Storici Paola, Zaliani Andrea

Optimization and Evaluation of Complementary Degrader Discovery Assays for Application in Screening.

优化和评价互补降解剂发现试验在筛选中的应用

Huchting Johanna, Weller Arjen, Schweizer Moyra, Brandt Mona, Heering Jan, Kuzikov Maria, Wolf Markus, Reinshagen Jeanette, Queisser Markus A, Gribbon Philip, Zaliani Andrea, Pless Ole, Kannt Aimo

From library to landscape: integrative annotation workflows for compound libraries in drug repurposing

从库到景观:药物重定位中化合物库的整合注释工作流程

Reinshagen, Jeanette; Seashore-Ludlow, Brinton; Gadiya, Yojana; Gustavsson, Anna-Lena; Tanoli, Ziaurrehman; Aittokallio, Tero; Huchting, Johanna; Jenmalm-Jensen, Annika; Gribbon, Philip; Zaliani, Andrea; Ballante, Flavio