日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting N-Myc in neuroblastoma with selective Aurora kinase A degraders.

利用选择性 Aurora 激酶 A 降解剂靶向神经母细胞瘤中的 N-Myc

Tang Jian, Moorthy Ramkumar, Hirsch Laura E, Demir Özlem, Baker Zachary D, Naumann Jordan A, Jones Katherine F M, Grillo Michael J, Haefner Ella S, Shi Ke, Levy Michaella J, Gupta Harshita B, Aihara Hideki, Harris Reuben S, Amaro Rommie E, Levinson Nicholas M, Harki Daniel A

Fragment-Based NMR Screening of the BPTF PHD Finger Methyl Lysine Reader Leads to the First Small-Molecule Inhibitors

基于片段的 NMR 筛选 BPTF PHD 指状甲基赖氨酸读取蛋白,发现了首批小分子抑制剂

Buchholz, Caroline R; Sneddon, Molly S; McPherson, Joseph E; Das, Sourav; Gee, Clifford T; Grillo, Michael J; Chai, Sergio C; Lee, Richard E; Chen, Taosheng; Harki, Daniel A; Shelat, Anang A; Pomerantz, William C K

The current toolbox for APOBEC drug discovery

APOBEC药物发现的现有工具箱

Grillo, Michael J; Jones, Katherine F M; Carpenter, Michael A; Harris, Reuben S; Harki, Daniel A

Case report of apoptosis in testis of four AZFc-deleted patients: increased DNA fragmentation during meiosis, but decreased apoptotic markers in post-meiotic germ cells

四例AZFc缺失患者睾丸细胞凋亡病例报告:减数分裂期间DNA碎片增加,但减数分裂后生殖细胞凋亡标志物减少

Eric Streichemberger, Jeanne Perrin, Jacqueline Saias-Magnan, Gilles Karsenty, Perrine Malzac, Jean-Marie Grillo, Michael J Mitchell, Catherine Metzler-Guillemain