日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Reducing hERG Inhibition in the Design of Potent and Bioavailable Indazole cGAS Inhibitors

在设计高效且生物利用度高的吲唑类cGAS抑制剂时降低hERG抑制

Cyr, Patrick; Chefson, Amandine; Sietsema, Daniel V; Konteatis, Zenon; Ciblat, Stéphane; Sgarioto, Nicolas; Le Gros, Philippe; Pike, Kelly A; Boily, Marc-Olivier; Diallo, Mohamed; Seliniotakis, Ria; Springer, Clayton; Khandelwal, Pradhyum; Beveridge, Ramsay E

Type I interferon-dependent and -independent signaling underlie autoantibody production in a murine lupus model.

I 型干扰素依赖性和非依赖性信号传导是小鼠狼疮模型中自身抗体产生的基础。

Levine Jerrold S, Pilon Céleste, Subang Rebecca, Salem David, Lonina Elena, Qureshi Salman T, Fonseca Gregory J, Gros Philippe, Rauch Joyce

Femtosecond Infrared Spectroscopy Resolving the Multiplicity of High-Spin Crossover States in Transition Metal Iron Complexes

飞秒红外光谱解析过渡金属铁配合物中高自旋交叉态的多重性

Zahn, Clark; Pastore, Mariachiara; Lustres, J Luis Perez; Gros, Philippe C; Haacke, Stefan; Heyne, Karsten

The potential importance of the built-environment microbiome and its impact on human health

建筑环境微生物组的潜在重要性及其对人类健康的影响

Bosch, Thomas C G; Wigley, Mark; Colomina, Beatriz; Bohannan, Brendan; Meggers, Forrest; Amato, Katherine R; Azad, Meghan B; Blaser, Martin J; Brown, Kate; Dominguez-Bello, Maria Gloria; Ehrlich, Stanislav Dusko; Elinav, Eran; Finlay, B Brett; Geddie, Kate; Geva-Zatorsky, Naama; Giles-Vernick, Tamara; Gros, Philippe; Guillemin, Karen; Haraoui, Louis-Patrick; Johnson, Elizabeth; Keck, Frédéric; Lorimer, Jamie; McFall-Ngai, Margaret J; Nichter, Mark; Pettersson, Sven; Poinar, Hendrik; Rees, Tobias; Tropini, Carolina; Undurraga, Eduardo A; Zhao, Liping; Melby, Melissa K

Discovery of Potent and Orally Bioavailable Pyrimidine Amide cGAS Inhibitors via Structure-Guided Hybridization

通过结构导向杂交发现高效且口服生物利用度高的嘧啶酰胺类cGAS抑制剂

Cyr, Patrick; Fader, Lee D; Burch, Jason D; Pike, Kelly A; Sietsema, Daniel V; Boily, Marc-Olivier; Ciblat, Stéphane; Sgarioto, Nicolas; Skeldon, Alexander M; Gaudreault, Samuel; Le Gros, Philippe; Dumais, Valérie; McKay, Daniel J J; Abraham, Nathan S; Seliniotakis, Ria; Beveridge, Ramsay E

Panchromatic light harvesting and record power conversion efficiency for carboxylic/cyanoacrylic Fe(ii) NHC co-sensitized FeSSCs

羧基/氰基丙烯酸酯Fe(II) NHC共敏化FeSSC的全色光捕获和创纪录的功率转换效率

Reddy-Marri, Anil; Marchini, Edoardo; Cabanes, Valentin Diez; Argazzi, Roberto; Pastore, Mariachiara; Caramori, Stefano; Gros, Philippe C

Case report: Diagnosis, management and evolution of a bulky and invasive cardiac mass complicated by complete atrioventricular block

病例报告:巨大且侵袭性心脏肿块合并完全性房室传导阻滞的诊断、治疗及演变。

Bohbot, Yohann; Garot, Jérôme; Danjon, Isabelle; Thébert, Dominique; Nahory, Louis; Gros, Philippe; Salerno, Fiorella; Garot, Philippe

Inherited human c-Rel deficiency disrupts myeloid and lymphoid immunity to multiple infectious agents

遗传性人类c-Rel缺乏症会破坏髓系和淋巴系对多种感染性病原体的免疫力。

Lévy, Romain; Langlais, David; Béziat, Vivien; Rapaport, Franck; Rao, Geetha; Lazarov, Tomi; Bourgey, Mathieu; Zhou, Yu J; Briand, Coralie; Moriya, Kunihiko; Ailal, Fatima; Avery, Danielle T; Markle, Janet; Lim, Ai Ing; Ogishi, Masato; Yang, Rui; Pelham, Simon; Emam, Mehdi; Migaud, Mélanie; Deswarte, Caroline; Habib, Tanwir; Saraiva, Luis R; Moussa, Eman A; Guennoun, Andrea; Boisson, Bertrand; Belkaya, Serkan; Martinez-Barricarte, Ruben; Rosain, Jérémie; Belkadi, Aziz; Breton, Sylvain; Payne, Kathryn; Benhsaien, Ibtihal; Plebani, Alessandro; Lougaris, Vassilios; Di Santo, James P; Neven, Bénédicte; Abel, Laurent; Ma, Cindy S; Bousfiha, Ahmed Aziz; Marr, Nico; Bustamante, Jacinta; Liu, Kang; Gros, Philippe; Geissmann, Frédéric; Tangye, Stuart G; Casanova, Jean-Laurent; Puel, Anne

The hygiene hypothesis, the COVID pandemic, and consequences for the human microbiome

卫生假说、新冠疫情及其对人类微生物组的影响

Finlay, B Brett; Amato, Katherine R; Azad, Meghan; Blaser, Martin J; Bosch, Thomas C G; Chu, Hiutung; Dominguez-Bello, Maria Gloria; Ehrlich, Stanislav Dusko; Elinav, Eran; Geva-Zatorsky, Naama; Gros, Philippe; Guillemin, Karen; Keck, Frédéric; Korem, Tal; McFall-Ngai, Margaret J; Melby, Melissa K; Nichter, Mark; Pettersson, Sven; Poinar, Hendrik; Rees, Tobias; Tropini, Carolina; Zhao, Liping; Giles-Vernick, Tamara

Tuneable access to indole, indolone, and cinnoline derivatives from a common 1,4-diketone Michael acceptor

通过常见的1,4-二酮迈克尔受体,可调控地合成吲哚、吲哚酮和噌啉衍生物

El-Marrouki, Dalel; Touchet, Sabrina; Abdelli, Abderrahmen; M'Rabet, Hédi; Lotfi Efrit, Mohamed; Gros, Philippe C