日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure guided modification of 2-chloro-5-(ethyl-phenyl-sulfamoyl)-N-[2-(2-oxo-pyrrolidin-1-yl)-phenyl]-benzamide to afford selective inhibitors of Cryptosporidium parvum N-myristoyltransferase

以2-氯-5-(乙基苯基磺酰基)-N-[2-(2-氧代吡咯烷-1-基)苯基]-苯甲酰胺为模板,构建选择性小隐孢子虫N-肉豆蔻酰转移酶抑制剂

Sigalapalli, Dilep K; Groustra, Sophia; Fenwick, Michael K; Zigweid, Rachael; Hulverson, Matthew A; Owsley, Eric; Khim, Monique; Shibata, Sayaka; Van Voorhis, Wesley C; Staker, Bart L; Fan, Erkang

Selective Bias Virtual Screening for Discovery of Promising Antimalarial Candidates targeting Plasmodium N-Myristoyltransferase

利用选择性偏倚虚拟筛选发现靶向疟原虫N-肉豆蔻酰转移酶的潜在抗疟候选药物

Andrade, Carolina; Sousa, Bruna Katiele de Paula; Sigurdardóttir, Sunniva; Bourgard, Catarina; Borba, Joyce; Clementino, Leandro; Salazar-Alvarez, Luis Carlos; Groustra, Sophia; Zigweid, Rachael; Khim, Monique; Staker, Bart; Costa, Fabio; Eriksson, Leif; Sunnerhagen, Per