日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Elucidating Compound Mechanism of Action and Polypharmacology with a Large-scale Perturbational Profile Compendium

利用大规模扰动谱汇编阐明化合物的作用机制和多药理学

Hu, Lucas ZhongMing; Hirschhorn, Tal; Douglass, Eugene; Murray, Diana; Trudeau, Stephen J; Turunen, Mikko; Pampou, Sergey; Grunn, Adina; Realubit, Ron; Antolin, Albert A; Wang, Alexander L E; Li, Hai; Subramaniam, Prem; Mundi, Prabhjot S; Karan, Charles; Alvarez, Mariano; Honig, Barry; Stockwell, Brent R; Califano, Andrea

Identification and Pharmacological Targeting of Treatment-Resistant, Stem-like Breast Cancer Cells for Combination Therapy

识别和药理学靶向治疗耐药性干细胞样乳腺癌细胞以进行联合治疗

Jeremy Worley, Heeju Noh, Daoqi You, Mikko M Turunen, Hongxu Ding, Evan Paull, Aaron T Griffin, Adina Grunn, Mingxuan Zhang, Kristina Guillan, Erin C Bush, Samantha J Brosius, Hanina Hibshoosh, Prabhjot S Mundi, Peter Sims, Piero Dalerba, Filemon S Dela Cruz, Andrew L Kung, Andrea Califano

Systematic elucidation and pharmacologic targeting on non-oncogene dependencies in imatinib-resistant gastrointestinal stromal tumor

系统阐明和药物靶向治疗伊马替尼耐药性胃肠道间质瘤中的非癌基因依赖性

Mundi, Prabhjot S; Grunn, Adina; Kojadinovic, Arsenije; Karan, Charles; Realubit, Ronald; Caescu, Cristina I; Hibshoosh, Hanina; Aburi, Mahalaxmi; Alvarez, Mariano J; Ingham, Matthew; Evans, Denisse; Rothschild, Sara; Schwartz, Gary K; Califano, Andrea

A Transcriptome-Based Precision Oncology Platform for Patient-Therapy Alignment in a Diverse Set of Treatment-Resistant Malignancies.

基于转录组的精准肿瘤学平台,用于针对多种难治性恶性肿瘤的患者-治疗方案匹配

Mundi Prabhjot S, Dela Cruz Filemon S, Grunn Adina, Diolaiti Daniel, Mauguen Audrey, Rainey Allison R, Guillan Kristina, Siddiquee Armaan, You Daoqi, Realubit Ronald, Karan Charles, Ortiz Michael V, Douglass Eugene F, Accordino Melissa, Mistretta Suzanne, Brogan Frances, Bruce Jeffrey N, Caescu Cristina I, Carvajal Richard D, Crew Katherine D, Decastro Guarionex, Heaney Mark, Henick Brian S, Hershman Dawn L, Hou June Y, Iwamoto Fabio M, Jurcic Joseph G, Kiran Ravi P, Kluger Michael D, Kreisl Teri, Lamanna Nicole, Lassman Andrew B, Lim Emerson A, Manji Gulam A, McKhann Guy M, McKiernan James M, Neugut Alfred I, Olive Kenneth P, Rosenblat Todd, Schwartz Gary K, Shu Catherine A, Sisti Michael B, Tergas Ana, Vattakalam Reena M, Welch Mary, Wenske Sven, Wright Jason D, Canoll Peter, Hibshoosh Hanina, Kalinsky Kevin, Aburi Mahalaxmi, Sims Peter A, Alvarez Mariano J, Kung Andrew L, Califano Andrea

Validation of a non-oncogene encoded vulnerability to exportin 1 inhibition in pediatric renal tumors

验证儿童肾肿瘤中非癌基因编码的对输出蛋白1抑制剂的易感性

Diego F Coutinho ,Prabhjot S Mundi ,Lianna J Marks ,Chelsey Burke ,Michael V Ortiz ,Daniel Diolaiti ,Lauren Bird ,Kelly L Vallance ,Glorymar Ibáñez ,Daoqi You ,Matthew Long ,Nestor Rosales ,Adina Grunn ,Andoyo Ndengu ,Armaan Siddiquee ,Ervin S Gaviria ,Allison R Rainey ,Ladan Fazlollahi ,Hajime Hosoi ,Andrea Califano ,Andrew L Kung ,Filemon S Dela Cruz

A precision oncology approach to the pharmacological targeting of mechanistic dependencies in neuroendocrine tumors

精准肿瘤学方法在神经内分泌肿瘤机制依赖性药物靶向治疗中的应用

Alvarez, Mariano J; Subramaniam, Prem S; Tang, Laura H; Grunn, Adina; Aburi, Mahalaxmi; Rieckhof, Gabrielle; Komissarova, Elena V; Hagan, Elizabeth A; Bodei, Lisa; Clemons, Paul A; Dela Cruz, Filemon S; Dhall, Deepti; Diolaiti, Daniel; Fraker, Douglas A; Ghavami, Afshin; Kaemmerer, Daniel; Karan, Charles; Kidd, Mark; Kim, Kyoung M; Kim, Hee C; Kunju, Lakshmi P; Langel, Ülo; Li, Zhong; Lee, Jeeyun; Li, Hai; LiVolsi, Virginia; Pfragner, Roswitha; Rainey, Allison R; Realubit, Ronald B; Remotti, Helen; Regberg, Jakob; Roses, Robert; Rustgi, Anil; Sepulveda, Antonia R; Serra, Stefano; Shi, Chanjuan; Yuan, Xiaopu; Barberis, Massimo; Bergamaschi, Roberto; Chinnaiyan, Arul M; Detre, Tony; Ezzat, Shereen; Frilling, Andrea; Hommann, Merten; Jaeger, Dirk; Kim, Michelle K; Knudsen, Beatrice S; Kung, Andrew L; Leahy, Emer; Metz, David C; Milsom, Jeffrey W; Park, Young S; Reidy-Lagunes, Diane; Schreiber, Stuart; Washington, Kay; Wiedenmann, Bertram; Modlin, Irvin; Califano, Andrea

Inactivating mutations of acetyltransferase genes in B-cell lymphoma

细胞淋巴瘤中乙酰转移酶基因的失活突变

Laura Pasqualucci, David Dominguez-Sola, Annalisa Chiarenza, Giulia Fabbri, Adina Grunn, Vladimir Trifonov, Lawryn H Kasper, Stephanie Lerach, Hongyan Tang, Jing Ma, Davide Rossi, Amy Chadburn, Vundavalli V Murty, Charles G Mullighan, Gianluca Gaidano, Raul Rabadan, Paul K Brindle, Riccardo Dalla-Fa

Mutations of multiple genes cause deregulation of NF-kappaB in diffuse large B-cell lymphoma

弥漫性大B细胞淋巴瘤中多个基因的突变导致NF-κB失调

Compagno, Mara; Lim, Wei Keat; Grunn, Adina; Nandula, Subhadra V; Brahmachary, Manisha; Shen, Qiong; Bertoni, Francesco; Ponzoni, Maurilio; Scandurra, Marta; Califano, Andrea; Bhagat, Govind; Chadburn, Amy; Dalla-Favera, Riccardo; Pasqualucci, Laura

Inactivation of the PRDM1/BLIMP1 gene in diffuse large B cell lymphoma

弥漫性大B细胞淋巴瘤中PRDM1/BLIMP1基因的失活

Pasqualucci, Laura; Compagno, Mara; Houldsworth, Jane; Monti, Stefano; Grunn, Adina; Nandula, Subhadra V; Aster, Jon C; Murty, Vundavally V; Shipp, Margaret A; Dalla-Favera, Riccardo

A genomewide screen of 345 families for autism-susceptibility loci

对345个家庭进行全基因组自闭症易感基因位点筛查

Yonan, Amanda L; Alarcón, Maricela; Cheng, Rong; Magnusson, Patrik K E; Spence, Sarah J; Palmer, Abraham A; Grunn, Adina; Juo, Suh-Hang Hank; Terwilliger, Joseph D; Liu, Jianjun; Cantor, Rita M; Geschwind, Daniel H; Gilliam, T Conrad