Single-position ligand modifications tune CB(2)R activity by targeting the toggle switch
通过靶向开关,单点配体修饰可以调节 CB(2)R 的活性。
期刊:Chemical Science
影响因子:7.4
doi:10.1039/d6sc00062b
Ganzoni, Rudolf L Z; Kosar, Miroslav; Han, Yongqi; Vitale, Rosa Maria; Amodeo, Pietro; Li, Xiaoting; Zha, Zhonghua; Patej, Kacper J; Kicin, Bilal; Strunden, Taddäus E N; Reichert, Lisa; Gómez-Bouzó, Uxía; Perera, Themiya P; Atz, Kenneth; Guba, Wolfgang; Bartelmus, Christian; Bigler, Raphael; Tosatti, Paolo; Bachmann, Stephan; Hua, Tian; Sykes, David A; Veprintsev, Dmitry B; Grether, Uwe; Carreira, Erick M