Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity.
发现 CLPP-1071 是一种效力极强、口服有效的 ClpP 激活剂,具有强大的体内抗肿瘤活性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c01605
Chen Beijing, Sun Mingyang, Zhang Chun, Huang Qi, Teng Dan, Hu Linghao, Ma Huicong, Lin Xinyi, Huang Zan, Gui Renzhao, Hu Xiaobei, Xu Lei, Zheng Mingyue, Zhou Yubo, Li Jia, Wang Mingliang