日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oxyprenyl-chalcones as antibacterial hits: design of experiments-optimized synthesis, antibacterial evaluation, early drug-like profiling and biodegradability prediction

氧异戊烯基查尔酮类化合物作为抗菌先导化合物:实验设计优化合成、抗菌活性评价、早期类药性分析和生物降解性预测

Marotta, Ludovica; Giammarino, Francesca Maria Pia Rita; Senenou Tambou, Brondon Brandly; Tudino, Valeria; Butini, Stefania; Broccardo, Lorenza; Cancade, Sacha Michèle Idriss; Docquier, Jean-Denis; Perego, Federica; Basilico, Nicoletta; Raffellini, Lorenzo; Gul, Sheraz; Carullo, Gabriele; Gemma, Sandra; Campiani, Giuseppe

Single-cell insights into tumor microenvironment heterogeneity and plasticity: transforming precision therapy in gastrointestinal cancers

单细胞视角揭示肿瘤微环境异质性和可塑性:革新胃肠道癌症的精准治疗

Weng, Jialei; Ju, Feng; Lyu, Zicheng; Fan, Ningbo; Smit, Daniel J; Xu, Wenxin; Wu, Xiaolin; Becker, Philip; Xu, Yinan; Schweiger, Michal R; Hillmer, Axel M; Harwig, Ralf; Gul, Sheraz; Link, Alexander; Meder, Lydia; Fang, Nan; Dong, Qiongzhu; Bruns, Christiane J; Ren, Ning; Zhao, Yue

Serial-femtosecond crystallography reveals how a phytochrome variant couples chromophore and protein structural changes

连续飞秒晶体学揭示了植物光敏色素变体如何耦合发色团和蛋白质的结构变化

Sauthof, Luisa; Szczepek, Michal; Schmidt, Andrea; Bhowmick, Asmit; Dasgupta, Medhanjali; Mackintosh, Megan J; Gul, Sheraz; Fuller, Franklin D; Chatterjee, Ruchira; Young, Iris D; Michael, Norbert; Heyder, Nicolas Andreas; Bauer, Brian; Koch, Anja; Bogacz, Isabel; Kim, In-Sik; Simon, Philipp S; Butryn, Agata; Aller, Pierre; Chukhutsina, Volha U; Baxter, James M; Hutchison, Christopher D M; Liebschner, Dorothee; Poon, Billy; Sauter, Nicholas K; Miller, Mitchell D; George N Phillips Jr; Alonso-Mori, Roberto; Hunter, Mark S; Batyuk, Alexander; Owada, Shigeki; Tono, Kensuke; Tanaka, Rie; van Thor, Jasper J; Krauß, Norbert; Lamparter, Tilman; Brewster, Aaron S; Schapiro, Igor; Orville, Allen M; Yachandra, Vittal K; Yano, Junko; Hildebrandt, Peter; Kern, Jan F; Scheerer, Patrick

Design of 2-Aminobenzothiazole Derivatives Targeting Trypanosomatid PTR1 by a Multidisciplinary Fragment Hybridization Approach

利用多学科片段杂交方法设计靶向锥虫 PTR1 的 2-氨基苯并噻唑衍生物

Panecka-Hofman, Joanna; Linciano, Pasquale; Pöhner, Ina; Dyguda-Kazimierowicz, Edyta; Jedwabny, Wiktoria; Landi, Giacomo; Santarem, Nuno; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Luciani, Rosaria; Ferrari, Stefania; Aiello, Daniele; Mangani, Stefano; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Costi, Maria Paola; Wade, Rebecca C

IGF2BP1-HAX-1 positive feedback loop-mediated HAX-1 overexpression blocks autophagic flux and promotes chemoresistance in nasopharyngeal carcinoma.

IGF2BP1-HAX-1 正反馈环介导的 HAX-1 过表达阻断自噬通量,促进鼻咽癌的化疗耐药性

Zhang Siyu, Gu Miao, Yin Haimeng, Pan Si, Xie Haijing, Chen Wenhui, Gul Sheraz, Zhao Yue, Wang Zhefang, Zheng Wenjie, You Yiwen, You Bo

Changes in metabolism-related RNA expression in circulating white blood cells of aged individual with physical frailty

老年体弱者循环白细胞中代谢相关RNA表达的变化

Okinaka, Yuka; Suda, Yoshihito; Matsumoto, Tomoyuki; Kuroda, Ryosuke; Shinagawa, Yoshiyuki; Gul, Sheraz; Claussen, Carsten; Matsui, Ikuko; Matsui, Yutaka; Taguchi, Akihiko

Design, synthesis and evaluation of pyrimidinobenzylamide and pyrimidinothiophenamide derivatives as inhibitors of DOT1L and related epigenetic targets DNMT3a, PRMT4 and other HMTs

设计、合成和评价嘧啶并苄酰胺和嘧啶并噻吩酰胺衍生物作为DOT1L及相关表观遗传靶点DNMT3a、PRMT4和其他HMTs的抑制剂

Castillo-Aguilera, Oscar Omar; Depreux, Patrick; Halby, Ludovic; Bailly, Christian; Domínguez-Ramírez, Lenin; Gul, Sheraz; Arimondo, Paola B; Goossens, Laurence

SAR Study of 4,8-Disubstituted Pyrimido[5,4-d]pyrimidines Exhibiting Antitrypanosomal and Antileishmanial Activity

4,8-二取代嘧啶并[5,4-d]嘧啶类化合物的构效关系研究及其抗锥虫和抗利什曼原虫活性

Lopes, André; Teixeira, Sofia; Santarém, Nuno; Greco, Alessandro; Pagliaro, Angela; Keminer, Oliver; Gul, Sheraz; Cordeiro-da-Silva, Anabela; Carvalho, Maria Alice

RNA Analysis of Circulating Leukocytes in Patients with Alzheimer's Disease

阿尔茨海默病患者循环白细胞的RNA分析

Okinaka, Yuka; Shinagawa, Yoshiyuki; Claussen, Carsten; Gul, Sheraz; Matsui, Ikuko; Matsui, Yutaka; Taguchi, Akihiko

In-vitro Cytotoxicity Investigations for Phytoconstituents of Saudi Medicinal Plants With Putative Ocular Effects

沙特阿拉伯药用植物中具有潜在眼部作用的植物成分的体外细胞毒性研究

Alghamdi, Ali Hendi; Ahmed, Aimun A E; Abdalgadir, Haidar; Bashir, Mahadi; Khalid, Asaad; Abdalla, Ashraf N; Elzubier, Mohamed E; Adnan Almaimani, Riyad; Refaat, Bassem; Alzahrani, Khalid; Alghamdi, Saleh M S; Gul, Sheraz