日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Histone decrotonylation plays a distinct role in HIV latency

组蛋白去泛素化在HIV潜伏期中发挥着独特的作用

Li, Xiaoyi; Li, Dajiang; Tang, Yuyang; Nearing, Marie; Varco-Merth, Benjamin; Chen, Hongjie; Smith, Davey; Gianella, Sara; Archin, Nancie M; Okoye, Afam A; Dandekar, Satya; Margolis, David M; Chirasani, Venkat R; Gumpper, Ryan H; Jiang, Guochun

Structural insights into coffee bitter taste perception by TAS2R43 receptor

TAS2R43受体对咖啡苦味感知的结构性见解

Kim, Yoojoong; Gumpper, Ryan H; Zhuang, Yuxuan; Dror, Ron O; Roth, Bryan L

Pan-Cancer Analysis Identifies a Ras-Related GTPase as a Potential Modulator of Cancer

泛癌分析发现Ras相关GTP酶可能是癌症的潜在调节因子。

Hsueh, Hsiang-Yin; Gumpper-Fedus, Kristyn; Poelstra, Jelmer W; Pitter, Kenneth L; Cruz-Monserrate, Zobeida

Molecular Glues: A New Approach to Modulating GPCR Signaling Bias

分子胶:一种调节GPCR信号偏向的新方法

Kushnir, Jamie; Gumpper, Ryan H

Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Michael Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Clinical risk factors for sarcopenia in acute and chronic pancreatitis

急性和慢性胰腺炎患者肌少症的临床危险因素

Ramsey, Mitchell L; Lu, Andrew; Gumpper-Fedus, Kristyn; Culp, Stacey; Bradley, David; Conwell, Darwin L; Cruz-Monserrate, Zobeida; Groce, J Royce; Han, Samuel; Krishna, Somashekar G; Lee, Peter; Mace, Thomas; Papachristou, Georgios I; Roberts, Kristen M; Shah, Zarine K; Hart, Phil A

Differential effects of sodium on agonist-induced conformational transitions and signaling at μ and κ opioid receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma M; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Ketogenic diet prevents obesity-associated pancreatic cancer independent of weight loss and induces pancreatic metabolic reprogramming.

生酮饮食可以预防与肥胖相关的胰腺癌,而无需减肥,并能诱导胰腺代谢重编程

Vélez-Bonet Ericka, Gumpper-Fedus Kristyn, Chasser Kaylin, Hurst Zachary, Hsueh Hsiang-Yin, Pita-Grisanti Valentina, Liette Alexus, Vulic Grace, Choueiry Fouad, Zhang Huan, Zhu Jiangjiang, Knoblaugh Sue E, Culp Stacey, Volek Jeff S, Cruz-Monserrate Zobeida

AlphaFold2 structures guide prospective ligand discovery

AlphaFold2结构指导潜在配体的发现

Lyu, Jiankun; Kapolka, Nicholas; Gumpper, Ryan; Alon, Assaf; Wang, Liang; Jain, Manish K; Barros-Álvarez, Ximena; Sakamoto, Kensuke; Kim, Yoojoong; DiBerto, Jeffrey; Kim, Kuglae; Glenn, Isabella S; Tummino, Tia A; Huang, Sijie; Irwin, John J; Tarkhanova, Olga O; Moroz, Yurii; Skiniotis, Georgios; Kruse, Andrew C; Shoichet, Brian K; Roth, Bryan L

Structure-guided design of a peripherally restricted chemogenetic system.

结构导向的外周限制性化学遗传系统设计

Kang Hye Jin, Krumm Brian E, Tassou Adrien, Geron Matan, DiBerto Jeffrey F, Kapolka Nicholas J, Gumpper Ryan H, Sakamoto Kensuke, Dewran Kocak D, Olsen Reid H J, Huang Xi-Ping, Zhang Shicheng, Huang Karen L, Zaidi Saheem A, Nguyen MyV T, Jo Min Jeong, Katritch Vsevolod, Fay Jonathan F, Scherrer Grégory, Roth Bryan L