日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Histone decrotonylation plays a distinct role in HIV latency

组蛋白去泛素化在HIV潜伏期中发挥着独特的作用

Li, Xiaoyi; Li, Dajiang; Tang, Yuyang; Nearing, Marie; Varco-Merth, Benjamin; Chen, Hongjie; Smith, Davey; Gianella, Sara; Archin, Nancie M; Okoye, Afam A; Dandekar, Satya; Margolis, David M; Chirasani, Venkat R; Gumpper, Ryan H; Jiang, Guochun

Structural insights into coffee bitter taste perception by TAS2R43 receptor

TAS2R43受体对咖啡苦味感知的结构性见解

Kim, Yoojoong; Gumpper, Ryan H; Zhuang, Yuxuan; Dror, Ron O; Roth, Bryan L

The structural diversity of psychedelic drug actions revealed

迷幻药作用的结构多样性揭示

Gumpper, Ryan H; Jain, Manish K; Kim, Kuglae; Sun, Renhong; Sun, Ning; Xu, Zhongli; DiBerto, Jeffrey F; Krumm, Brian E; Kapolka, Nicholas J; Kaniskan, H Ümit; Nichols, David E; Jin, Jian; Fay, Jonathan F; Roth, Bryan L

Molecular Glues: A New Approach to Modulating GPCR Signaling Bias

分子胶:一种调节GPCR信号偏向的新方法

Kushnir, Jamie; Gumpper, Ryan H

Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Michael Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Differential effects of sodium on agonist-induced conformational transitions and signaling at μ and κ opioid receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma M; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Structure-guided design of a peripherally restricted chemogenetic system.

结构导向的外周限制性化学遗传系统设计

Kang Hye Jin, Krumm Brian E, Tassou Adrien, Geron Matan, DiBerto Jeffrey F, Kapolka Nicholas J, Gumpper Ryan H, Sakamoto Kensuke, Dewran Kocak D, Olsen Reid H J, Huang Xi-Ping, Zhang Shicheng, Huang Karen L, Zaidi Saheem A, Nguyen MyV T, Jo Min Jeong, Katritch Vsevolod, Fay Jonathan F, Scherrer Grégory, Roth Bryan L

Psychedelics: preclinical insights provide directions for future research

迷幻剂:临床前研究成果为未来研究指明方向

Gumpper, Ryan H; Roth, Bryan L

High-affinity agonists reveal recognition motifs for the MRGPRD GPCR.

高亲和力激动剂揭示了 MRGPRD GPCR 的识别基序

Wang Chunyu, Liu Yongfeng, Lanier Marion, Yeager Adam, Singh Isha, Gumpper Ryan H, Krumm Brian E, DeLeon Chelsea, Zhang Shicheng, Boehm Marcus, Pittner Richard, Baron Alain, Dvorak Lisa, Bacon Corinne, Shoichet Brian K, Martinborough Esther, Fay Jonathan F, Cao Can, Roth Bryan L

DNA selection by the master transcription factor PU.1

主转录因子PU.1对DNA的选择

Terrell, J Ross; Taylor, Samuel J; Schneider, Amelia L; Lu, Yue; Vernon, Tyler N; Xhani, Suela; Gumpper, Ryan H; Luo, Ming; Wilson, W David; Steidl, Ulrich; Poon, Gregory M K