日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Beyond monoclonal antibodies: constraints and the case for alternative PD-1/PD-L1-targeting formats

单克隆抗体之外:局限性及替代性PD-1/PD-L1靶向疗法的必要性

Porozova, Natalia O; Petukhova, Natalia V; Gureev, Maxim A; Moiseev, Ivan S; Eliseev, Igor E; Fedorova, Ludmila V; Porozov, Yuri B

3-(3-Azabicyclo[2, 2, 1]heptan-2-yl)-1,2,4-oxadiazoles as Novel Potent DPP-4 Inhibitors to Treat T2DM.

3-(3-氮杂双环[2, 2, 1]庚烷-2-基)-1,2,4-恶二唑作为治疗2型糖尿病的新型强效DPP-4抑制剂

Zinevich Tatiana V, Maslov Ivan O, Kirichenko Olga G, Shorshnev Sergey V, Gureev Maxim A, Dolgushin Fedor M, Porozov Yuri B, Trukhan Vladimir M

Application of Rational Design and Molecular Metadynamics for the Estimation of Changes in Trans-Splicing Efficiency during the Mutagenesis of Ssp DnaE Intein.

应用理性设计和分子元动力学来估计 Ssp DnaE 内含肽诱变过程中反式剪接效率的变化

Sabantsev Matvei O, Brovin Andrew N, Gureev Maxim A, Porozov Yuri B, Chuvpilo Sergey A, Karabelsky Alexander V

The Potential of Usnic-Acid-Based Thiazolo-Thiophenes as Inhibitors of the Main Protease of SARS-CoV-2 Viruses

基于地衣酸的噻唑并噻吩类化合物作为SARS-CoV-2病毒主蛋白酶抑制剂的潜力

Yarovaya, Olga I; Filimonov, Aleksandr S; Baev, Dmitriy S; Borisevich, Sophia S; Zaykovskaya, Anna V; Chirkova, Varvara Yu; Marenina, Mariya K; Meshkova, Yulia V; Belenkaya, Svetlana V; Shcherbakov, Dmitriy N; Gureev, Maxim A; Luzina, Olga A; Pyankov, Oleg V; Salakhutdinov, Nariman F; Khvostov, Mikhail V

In Vitro Study of Biological Activity of Tanacetum vulgare Extracts

菊蒿提取物生物活性的体外研究

Babich, Olga; Larina, Viktoria; Krol, Olesia; Ulrikh, Elena; Sukhikh, Stanislav; Gureev, Maxim A; Prosekov, Alexander; Ivanova, Svetlana

Novel 1,2,4-Triazole- and Tetrazole-Containing 4H-Thiopyrano[2,3-b]quinolines: Synthesis Based on the Thio-Michael/aza-Morita-Baylis-Hillman Tandem Reaction and Investigation of Antiviral Activity

新型含1,2,4-三唑和四唑的4H-噻吩并[2,3-b]喹啉:基于硫代迈克尔/氮杂森田-贝利斯-希尔曼串联反应的合成及其抗病毒活性研究

Khramchikhin, Andrey V; Skryl'nikova, Mariya A; Gureev, Maxim A; Zarubaev, Vladimir V; Esaulkova, Iana L; Ilyina, Polina A; Mammeri, Oussama Abdelhamid; Spiridonova, Dar'ya V; Porozov, Yuri B; Ostrovskii, Vladimir A

π-π Noncovalent Interaction Involving 1,2,4- and 1,3,4-Oxadiazole Systems: The Combined Experimental, Theoretical, and Database Study

涉及1,2,4-和1,3,4-噁二唑体系的π-π非共价相互作用:实验、理论和数据库的综合研究

Baykov, Sergey V; Mikherdov, Alexander S; Novikov, Alexander S; Geyl, Kirill K; Tarasenko, Marina V; Gureev, Maxim A; Boyarskiy, Vadim P

Comparative Study of the Steroidogenic Effects of Human Chorionic Gonadotropin and Thieno[2,3-D]pyrimidine-Based Allosteric Agonist of Luteinizing Hormone Receptor in Young Adult, Aging and Diabetic Male Rats

人绒毛膜促性腺激素与噻吩并[2,3-D]嘧啶类黄体生成素受体变构激动剂对青年、老年和糖尿病雄性大鼠类固醇生成作用的比较研究

Bakhtyukov, Andrey A; Derkach, Kira V; Gureev, Maxim A; Dar'in, Dmitry V; Sorokoumov, Viktor N; Romanova, Irina V; Morina, Irina Yu; Stepochkina, Anna M; Shpakov, Alexander O