日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Insights from aquaporin structures into drug-resistant sleeping sickness

从水通道蛋白结构中揭示耐药性昏睡病的机制

Matusevicius, Modestas; Corey, Robin A; Gragera, Marcos; Yamashita, Keitaro; Sprenger, Teresa; Ungogo, Marzuq; Blaza, James N; Castro-Hartmann, Pablo; Chirgadze, Dimitri Y; Chaitanya Vedithi, Sundeep; Afanasyev, Pavel; Melero, Roberto; Warshamanage, Rangana; Gusach, Anastasiia; Carazo, José-Maria; Carrington, Mark; Blundell, Tom; Murshudov, Garib N; Stansfeld, Phillip J; Sansom, Mark S P; De Koning, Harry P; Tate, Christopher G; Weyand, Simone

Structure of the G(q)-coupled adhesion receptor ADGRL4

G(q)偶联黏附受体ADGRL4的结构

Chen, Qingchao; Gusach, Anastasiia; Diamante, Aurora; Patel, Jayesh C; Edwards, Patricia C; Tate, Christopher G; Favara, David M

Molecular recognition of an odorant by the murine trace amine-associated receptor TAAR7f

小鼠痕量胺相关受体TAAR7f对气味分子的分子识别

Gusach, Anastasiia; Lee, Yang; Khoshgrudi, Armin Nikpour; Mukhaleva, Elizaveta; Ma, Ning; Koers, Eline J; Chen, Qingchao; Edwards, Patricia C; Huang, Fanglu; Kim, Jonathan; Mancia, Filippo; Veprintsev, Dmitry B; Vaidehi, Nagarajan; Weyand, Simone N; Tate, Christopher G

Sub-millisecond conformational dynamics of the A2A adenosine receptor revealed by single-molecule FRET

单分子 FRET 揭示 A2A 腺苷受体的亚毫秒构象动力学

Ivan Maslov, Oleksandr Volkov, Polina Khorn, Philipp Orekhov, Anastasiia Gusach, Pavel Kuzmichev, Andrey Gerasimov, Aleksandra Luginina, Quinten Coucke, Andrey Bogorodskiy, Valentin Gordeliy, Simon Wanninger, Anders Barth, Alexey Mishin, Johan Hofkens, Vadim Cherezov, Thomas Gensch, Jelle Hendrix, V

Structural diversity of leukotriene G-protein coupled receptors

白三烯G蛋白偶联受体的结构多样性

Luginina, Aleksandra; Gusach, Anastasiia; Lyapina, Elizaveta; Khorn, Polina; Safronova, Nadezda; Shevtsov, Mikhail; Dmitirieva, Daria; Dashevskii, Dmitrii; Kotova, Tatiana; Smirnova, Ekaterina; Borshchevskiy, Valentin; Cherezov, Vadim; Mishin, Alexey

Structural basis for receptor selectivity and inverse agonism in S1P5 receptors

S1P5 受体选择性和反向激动的结构基础

Elizaveta Lyapina #, Egor Marin #, Anastasiia Gusach #, Philipp Orekhov, Andrey Gerasimov, Aleksandra Luginina, Daniil Vakhrameev, Margarita Ergasheva, Margarita Kovaleva, Georgii Khusainov, Polina Khorn, Mikhail Shevtsov, Kirill Kovalev, Sergey Bukhdruker, Ivan Okhrimenko, Petr Popov, Hao Hu, Uwe W

Small-wedge synchrotron and serial XFEL datasets for Cysteinyl leukotriene GPCRs

半胱氨酰白三烯 GPCR 的小楔同步加速器和串行 XFEL 数据集

Egor Marin, Aleksandra Luginina, Anastasiia Gusach, Kirill Kovalev, Sergey Bukhdruker, Polina Khorn, Vitaly Polovinkin, Elizaveta Lyapina, Andrey Rogachev, Valentin Gordeliy, Alexey Mishin, Vadim Cherezov, Valentin Borshchevskiy5

Hydroxylation of Antitubercular Drug Candidate, SQ109, by Mycobacterial Cytochrome P450

分枝杆菌细胞色素 P450 对抗结核病候选药物 SQ109 的羟基化

Sergey Bukhdruker, Tatsiana Varaksa, Irina Grabovec, Egor Marin, Polina Shabunya, Maria Kadukova, Sergei Grudinin, Anton Kavaleuski, Anastasiia Gusach, Andrei Gilep, Valentin Borshchevskiy, Natallia Strushkevich

Structural basis of ligand selectivity and disease mutations in cysteinyl leukotriene receptors

半胱氨酰白三烯受体的配体选择性和疾病突变的结构基础

Anastasiia Gusach, Aleksandra Luginina, Egor Marin, Rebecca L Brouillette, Élie Besserer-Offroy, Jean-Michel Longpré, Andrii Ishchenko, Petr Popov, Nilkanth Patel, Taku Fujimoto, Toru Maruyama, Benjamin Stauch, Margarita Ergasheva, Daria Romanovskaia, Anastasiia Stepko, Kirill Kovalev, Mikhail Shevt

Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs

抗哮喘药物抑制半胱氨酰白三烯受体的结构机制

Aleksandra Luginina, Anastasiia Gusach, Egor Marin, Alexey Mishin, Rebecca Brouillette, Petr Popov, Anna Shiriaeva, Élie Besserer-Offroy, Jean-Michel Longpré, Elizaveta Lyapina, Andrii Ishchenko, Nilkanth Patel, Vitaly Polovinkin, Nadezhda Safronova, Andrey Bogorodskiy, Evelina Edelweiss, Hao Hu, Uw