日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery, Structure-Activity Relationship, and Functional Characterization of a Chromenopyrrole Series as Orthosteric Antagonists of GPR84

色烯吡咯系列化合物作为GPR84正构拮抗剂的发现、构效关系及功能表征

Malone, Michael A; Yin, Ruijing; Li, Yueming; Jenkins, Laura; Guseinov, Abdul-Akim; Marsango, Sara; Huggett, Mark; Huggett, Margaret; Boyle, Anna; Morrison, Angus; Tikhonova, Irina G; Milligan, Graeme; Jamieson, Andrew G

Steroid Recognition in Adhesion GPCRs: A Structural and Pharmacological Perspective

粘附 GPCR 中的类固醇识别:结构和药理学视角

Fleming, Bethany; Guseinov, Abdul-Akim; Tikhonova, Irina G; Milligan, Graeme; Perry-Hauser, Nicole A

Consistent supra-molecular motifs and different local symmetries in the structures of 2-amino-5-(4-fluoro-phen-yl)-1,3-thia-zole-4-carbaldehyde and 2-amino-5-(4-chloro-phen-yl)-1,3-thia-zole-4-carbaldehyde

2-氨基-5-(4-氟苯基)-1,3-噻唑-4-甲醛和2-氨基-5-(4-氯苯基)-1,3-噻唑-4-甲醛的结构中存在一致的超分子基序和不同的局部对称性

Guseinov, Firudin I; Afanaseva, Ksenia A; Gaidar, Sergey M; Pikina, Anna M; Akkurt, Mehmet; Aliyeva, Fargana S; Hasanov, Khudayar I; Belay, Alebel N

Mechanism of GPR84 allosteric modulation at a helix 8-proximate site

GPR84 在螺旋 8 近端位点的变构调节机制

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Zhou, Jingkai; Gossen, Fabian; Wang, Pinqi; Al Mahmud, Zobaer; Li, Yueming; Mahardhika, Andhika B; Muller, Christa E; Feng, Mingye; Russell, Angela J; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Allosteric modulation and biased signalling at free fatty acid receptor 2

游离脂肪酸受体 2 的变构调节和偏向性信号传导

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Valentini, Alice; Marsango, Sara; Schultz-Knudsen, Katrine; Ulven, Trond; Rexen Ulven, Elisabeth; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Comprehensive Investigation of the Commercial ELP-20 Electron-Beam Lithography Resist

对商用ELP-20电子束光刻胶的全面调查

Qairat, Meruert; Alzhanova, Aliya; Pshikov, Mustakhim; Nemkayeva, Renata; Guseinov, Nazim; Zaitsev, Sergey; Muratov, Mukhit

Sensitivity and Contrast Characterization of PMMA 950K Resist Under 30 keV Focused Ga(+) Ion Beam Exposure

PMMA 950K光刻胶在30 keV聚焦Ga(+)离子束曝光下的灵敏度和对比度特性

Muratov, Mukhit; Shabelnikova, Yana; Zaitsev, Sergey; Nemkayeva, Renata; Guseinov, Nazim

Crystal structure of 1-[(4-chloro-phen-yl)di-phenylyl-meth-yl]-3-(tri-fluoro-meth-yl)-1H-pyrazole

1-[(4-氯苯基)二苯基甲基]-3-(三氟甲基)-1H-吡唑的晶体结构

Guseinov, Firudin I; Afanaseva, Ksenia A; A Vil, Vera; Ugrak, Bogdan I; Samigullina, Aida I; Zangrando, Ennio; Belay, Alebel N

Syntheses, crystal structures, Hirshfeld surface analyses and crystal voids of 1-(4-bromo-phen-yl)-2,2-di-chloro-ethan-1-one and 2,2-di-bromo-1-(p-tol-yl)ethan-1-one

1-(4-溴苯基)-2,2-二氯乙酮和2,2-二溴-1-(对甲苯基)乙酮的合成、晶体结构、Hirshfeld表面分析和晶体空隙

Gurbanov, Atash V; Guseinov, Firudin I; Samigullina, Aida I; Hökelek, Tuncer; Hasanov, Khudayar I; Javadzade, Tahir A; Belay, Alebel N

Synthesis and structure of 6-bromo-2-(di-eth-oxymeth-yl)-2-hy-droxy-3-phenyl-2,3-di-hydro-1H-imidazo[1,2-a]pyridin-4-ium chloride aceto-nitrile monosolvate

6-溴-2-(二乙氧基甲基)-2-羟基-3-苯基-2,3-二氢-1H-咪唑并[1,2-a]吡啶-4-鎓氯化物乙腈单溶剂化物的合成与结构

Guseinov, Firudin I; Samigullina, Aida I; Hökelek, Tuncer; Hamidov, Sahil Z; Lasri, Jamal; Hasanov, Khudayar I; Javadzade, Tahir A; Belay, Alebel N