日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combinations of the azaquinazoline anti-Wolbachia agent, AWZ1066S, with benzimidazole anthelmintics synergise to mediate sub-seven-day sterilising and curative efficacies in experimental models of filariasis

抗沃尔巴克氏体药物AWZ1066S(一种氮杂喹唑啉类药物)与苯并咪唑类驱虫药联合使用,可产生协同作用,在丝虫病实验模型中于7天内达到灭菌和治愈效果。

Hegde, Shrilakshmi; Marriott, Amy E; Pionnier, Nicolas; Steven, Andrew; Bulman, Christina; Gunderson, Emma; Vogel, Ian; Koschel, Marianne; Ehrens, Alexandra; Lustigman, Sara; Voronin, Denis; Tricoche, Nancy; Hoerauf, Achim; Hübner, Marc P; Sakanari, Judy; Aljayyoussi, Ghaith; Gusovsky, Fabian; Dagley, Jessica; Hong, David W; O'Neill, Paul; Ward, Steven A; Taylor, Mark J; Turner, Joseph D

Vaccine-linked chemotherapy improves cardiac structure and function in a mouse model of chronic Chagas disease

疫苗联合化疗可改善慢性恰加斯病小鼠模型的心脏结构和功能

Jones, Kathryn M; Mangin, Elise N; Reynolds, Corey L; Villanueva, Liliana E; Cruz, Julio Vladimir; Versteeg, Leroy; Keegan, Brian; Kendricks, April; Pollet, Jeroen; Gusovsky, Fabian; Bottazzi, Maria Elena; Hotez, Peter J

Combining SJ733, an oral ATP4 inhibitor of Plasmodium falciparum, with the pharmacokinetic enhancer cobicistat: An innovative approach in antimalarial drug development

将口服的恶性疟原虫ATP4抑制剂SJ733与药代动力学增强剂cobicistat联合使用:抗疟药物研发领域的一种创新方法

Gaur, Aditya H; Panetta, John C; Smith, Amber M; Dallas, Ronald H; Freeman, Burgess B 3rd; Stewart, Tracy B; Tang, Li; John, Elizabeth; Branum, Kristen C; Patel, Nehali D; Ost, Shelley; Heine, Ryan N; Richardson, Julie L; Hammill, Jared T; Bebrevska, Lidiya; Gusovsky, Fabian; Maki, Noritsugu; Yanagi, Toshiharu; Flynn, Patricia M; McCarthy, James S; Chalon, Stephan; Guy, R Kiplin

Vaccine-linked chemotherapy with a low dose of benznidazole plus a bivalent recombinant protein vaccine prevents the development of cardiac fibrosis caused by Trypanosoma cruzi in chronically-infected BALB/c mice

低剂量苯硝唑联合二价重组蛋白疫苗的疫苗联用化疗可预防慢性感染克氏锥虫的BALB/c小鼠发生心脏纤维化。

Dzul-Huchim, Victor Manuel; Ramirez-Sierra, Maria Jesus; Martinez-Vega, Pedro Pablo; Rosado-Vallado, Miguel Enrique; Arana-Argaez, Victor Ermilo; Ortega-Lopez, Jaime; Gusovsky, Fabian; Dumonteil, Eric; Cruz-Chan, Julio Vladimir; Hotez, Peter; Bottazzi, María Elena; Villanueva-Lizama, Liliana Estefania

The Tuberculosis Drug Accelerator at year 10: what have we learned?

结核病药物加速计划实施10周年:我们学到了什么?

Aldridge, Bree B; Barros-Aguirre, David; Barry, Clifton E 3rd; Bates, Robert H; Berthel, Steven J; Boshoff, Helena I; Chibale, Kelly; Chu, Xin-Jie; Cooper, Christopher B; Dartois, Véronique; Duncan, Ken; Fotouhi, Nader; Gusovsky, Fabian; Hipskind, Philip A; Kempf, Dale J; Lelièvre, Joël; Lenaerts, Anne J; McNamara, Case W; Mizrahi, Valerie; Nathan, Carl; Olsen, David B; Parish, Tanya; Petrassi, H Michael; Pym, Alexander; Rhee, Kyu Y; Robertson, Gregory T; Rock, Jeremy Michael; Rubin, Eric J; Russell, Betsy; Russell, David G; Sacchettini, James C; Schnappinger, Dirk; Schrimpf, Michael; Upton, Anna M; Warner, Peter; Wyatt, Paul Graham; Yuan, Ying

Allosteric inhibitors of Mycobacterium tuberculosis tryptophan synthase

结核分枝杆菌色氨酸合成酶的变构抑制剂

Michalska, Karolina; Chang, Changsoo; Maltseva, Natalia I; Jedrzejczak, Robert; Robertson, Gregory T; Gusovsky, Fabian; McCarren, Patrick; Schreiber, Stuart L; Nag, Partha P; Joachimiak, Andrzej

Influenza "Trains" the Host for Enhanced Susceptibility to Secondary Bacterial Infection

流感会“训练”宿主,使其更容易受到继发性细菌感染。

Shirey, Kari Ann; Perkins, Darren J; Lai, Wendy; Zhang, Wei; Fernando, Lurds R; Gusovsky, Fabian; Blanco, Jorge C G; Vogel, Stefanie N

Vaccine-Linked Chemotherapy Improves Benznidazole Efficacy for Acute Chagas Disease

疫苗联合化疗可提高苯硝唑治疗急性恰加斯病的疗效

Jones, Kathryn; Versteeg, Leroy; Damania, Ashish; Keegan, Brian; Kendricks, April; Pollet, Jeroen; Cruz-Chan, Julio Vladimir; Gusovsky, Fabian; Hotez, Peter J; Bottazzi, Maria Elena

Diversity-oriented synthesis yields novel multistage antimalarial inhibitors.

多样性导向合成产生新型多阶段抗疟疾抑制剂

Kato Nobutaka, Comer Eamon, Sakata-Kato Tomoyo, Sharma Arvind, Sharma Manmohan, Maetani Micah, Bastien Jessica, Brancucci Nicolas M, Bittker Joshua A, Corey Victoria, Clarke David, Derbyshire Emily R, Dornan Gillian L, Duffy Sandra, Eckley Sean, Itoe Maurice A, Koolen Karin M J, Lewis Timothy A, Lui Ping S, Lukens Amanda K, Lund Emily, March Sandra, Meibalan Elamaran, Meier Bennett C, McPhail Jacob A, Mitasev Branko, Moss Eli L, Sayes Morgane, Van Gessel Yvonne, Wawer Mathias J, Yoshinaga Takashi, Zeeman Anne-Marie, Avery Vicky M, Bhatia Sangeeta N, Burke John E, Catteruccia Flaminia, Clardy Jon C, Clemons Paul A, Dechering Koen J, Duvall Jeremy R, Foley Michael A, Gusovsky Fabian, Kocken Clemens H M, Marti Matthias, Morningstar Marshall L, Munoz Benito, Neafsey Daniel E, Sharma Amit, Winzeler Elizabeth A, Wirth Dyann F, Scherer Christina A, Schreiber Stuart L