日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel paracellular marker based on ᴅ-dipeptide structure for highly sensitive quantification with UPLC-MS/MS for in vitro and in vivo blood-brain barrier permeability analysis

基于D-二肽结构的新型细胞旁路标志物,可通过UPLC-MS/MS进行高灵敏度定量分析,用于体外和体内血脑屏障通透性分析。

Bay, Cindy; Mühlberg, Eric; Uhl, Philipp; Stingl, Julia Carolin; Bajraktari-Sylejmani, Gzona; Burhenne, Jürgen; Weiss, Johanna; Sauter, Max

Ependymoma group-specific blood-brain barrier differences uncovered by a multi-omics approach.

通过多组学方法揭示室管膜瘤组特异性血脑屏障差异。

Sundheimer Julia K, Benzel Julia, Federico Aniello, Volz Stefanie, Knoll Maximilian, Statz Britta, Zheng Tuyu, Kmiecik Szymon W, Burhenne Jürgen, Bajraktari-Sylejmani Gzona, Scheuermann Sophia, King Anke, Müller Torsten, Hübner Jens-Martin, Kalxdorf Mathias, Peterziel Heike, Oehme Ina, Krijgsveld Jeroen, Seitz Christian M, Kool Marcel, Pfister Stefan M, Pajtler Kristian W, Maaß Kendra K

The "specific" P-glycoprotein inhibitor zosuquidar (LY335979) also weakly inhibits human organic cation transporters

“特异性”P-糖蛋白抑制剂佐苏奎达(LY335979)也对人有机阳离子转运体有微弱的抑制作用。

Bajraktari-Sylejmani, Gzona; Kamaraj, Rajamanikkam; Theile, Dirk; Pávek, Petr; Weiss, Johanna

In vitro evaluation of the reductive carbonyl idarubicin metabolism to evaluate inhibitors of the formation of cardiotoxic idarubicinol via carbonyl and aldo-keto reductases

体外评价还原羰基伊达比星代谢,以评估通过羰基和醛酮还原酶形成心脏毒性伊达比星醇的抑制剂

Gzona Bajraktari-Sylejmani, Julia Sophie Oster, Jürgen Burhenne, Walter Emil Haefeli, Max Sauter #, Johanna Weiss #

A Highly Sensitive UPLC-MS/MS Method for the Quantification of the Organic Cation Transporters' Mediated Metformin Uptake and Its Inhibition in Cells

用于定量分析有机阳离子转运体介导的二甲双胍摄取及其在细胞中抑制作用的高灵敏度UPLC-MS/MS方法

Bajraktari-Sylejmani, Gzona; Bay, Cindy; Gebauer, Lukas; Burhenne, Jürgen; Weiss, Johanna; Sauter, Max

Extracellular Vesicles as Surrogates for the Regulation of the Drug Transporters ABCC2 (MRP2) and ABCG2 (BCRP)

细胞外囊泡作为药物转运蛋白 ABCC2 (MRP2) 和 ABCG2 (BCRP) 的调节替代品

Juan Pablo Rigalli, Anna Gagliardi, Klara Diester, Gzona Bajraktari-Sylejmani, Antje Blank, Jürgen Burhenne, Alexander Lenard, Lars Werntz, Andrea Huppertz, Lena Münch, Janica Margrit Wendt, Max Sauter, Walter Emil Haefeli, Johanna Weiss

Extracellular Vesicles as Surrogates for Drug Metabolism and Clearance: Promise vs. Reality

细胞外囊泡作为药物代谢和清除的替代物:前景与现实

Gagliardi, Anna; Bajraktari-Sylejmani, Gzona; Barocelli, Elisabetta; Weiss, Johanna; Rigalli, Juan Pablo

Evaluation of PepT1 (SLC15A1) Substrate Characteristics of Therapeutic Cyclic Peptides

治疗性环肽的PepT1(SLC15A1)底物特性评估

Gzona Bajraktari-Sylejmani, Teresa von Linde, Jürgen Burhenne, Walter Emil Haefeli, Max Sauter, Johanna Weiss

Functional Characterization of the Solute Carrier LAT-1 (SLC7A5/SLC2A3) in Human Brain Capillary Endothelial Cells with Rapid UPLC-MS/MS Quantification of Intracellular Isotopically Labelled L-Leucine

利用快速 UPLC-MS/MS 定量分析细胞内同位素标记的 L-亮氨酸,对人脑毛细血管内皮细胞中的溶质载体 LAT-1 (SLC7A5/SLC2A3) 进行功能表征

Cindy Bay, Gzona Bajraktari-Sylejmani, Walter E Haefeli, Jürgen Burhenne, Johanna Weiss, Max Sauter

Rapid and Sensitive Quantification of Intracellular Glycyl-Sarcosine for Semi-High-Throughput Screening for Inhibitors of PEPT-1

快速灵敏地定量细胞内甘氨酰肌氨酸,用于半高通量筛选PEPT-1抑制剂

von Linde, Teresa; Bajraktari-Sylejmani, Gzona; Haefeli, Walter E; Burhenne, Jürgen; Weiss, Johanna; Sauter, Max