日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Author Correction: Structural insights into antagonist recognition by the vasopressin V2 receptor

作者更正:血管加压素V2受体拮抗剂识别的结构解析

Zhang, Tianwei; Liu, Hongli; You, Chongzhao; Zhang, Yixiao; Xu, Youwei; Pan, Benxun; Wu, Canrong; Jin, Sanshan; Yin, Yu-Ling; Wu, Kai; Chen, Yue; Sun, Hong; Si, Yuan; Tan, Yangxia; Yin, Wanchao; Xu, H Eric; Guo, Dong; Jiang, Yi

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Fusion Strategy of DNA-Encoded Libraries Drives Discovery of Allosteric Inhibitors of SARS-CoV‑2 RdRp

DNA编码文库的融合策略推动了SARS-CoV-2 RNA依赖性RNA聚合酶(RdRp)变构抑制剂的发现。

Li, Linjie; Wang, Xudong; Ding, Peiqi; Shen, Xuanjing; Hu, Hangchen; Wang, Xiaoxi; Jin, Rui; Wu, Xinyuan; Zhang, Yiwei; Lu, Weiwei; Yue, Jinfeng; Xu, H Eric; Yin, Wanchao; Xu, Yechun; Lu, Xiaojie

Cryo-EM structures of GPR75 reveal an occluded orthosteric pocket challenging conventional drug discovery paradigms for an anti-obesity target

GPR75的冷冻电镜结构揭示了一个封闭的正构口袋,这挑战了传统的抗肥胖靶点药物发现模式。

Zhu, Zi-Ning; You, Chong-Zhao; Yuan, Qing-Ning; Xu, Jiu-Yin; Gu, Zong-Yue; Huang, Zheng; Liu, Miao; Shan, Bei; Wang, James Jiqi; Hu, Wen; Wang, Kai; Yin, Wan-Chao; Xu, You-Wei; Xu, H Eric; Wu, Can-Rong

Decoding ligand recognition and constitutive activation of histamine H3 and H4 receptors.

解码组胺H3和H4受体的配体识别和组成性激活。

Jin San-Shan, Zhang Heng, Yan Jia-Hui, Wu Can-Rong, Cai Xiao-Qing, Wu Kai, Wang Ming-Wei, Xu H Eric, Yang De-Hua, Jiang Yi

Structural insight into GPR55 ligand recognition and G-protein coupling

GPR55配体识别和G蛋白偶联的结构解析

Xia, Ruixue; Yuan, Qingning; Wang, Na; Hou, Li; Abe, Junpei; Song, Jing; Ito, Yukishige; Xu, H Eric; He, Yuanzheng

Molecular mechanism of the arrestin-biased agonism of neurotensin receptor 1 by an intracellular allosteric modulator

细胞内变构调节剂介导的神经降压素受体1的阻遏蛋白偏向性激动作用的分子机制

Sun, Demeng; Li, Xiang; Yuan, Qingning; Wang, Yuanxia; Shi, Pan; Zhang, Huanhuan; Wang, Tao; Sun, Wenjing; Ling, Shenglong; Liu, Yuanchun; Lai, Jinglin; Xie, Wenqin; Yin, Wanchao; Liu, Lei; Xu, H Eric; Tian, Changlin

Author Correction: Structural and functional evidence that GPR30 is not a direct estrogen receptor

作者更正:结构和功能证据表明 GPR30 不是直接的雌激素受体

Liu, Heng; Guo, Shimeng; Dai, Antao; Xu, Peiyu; Li, Xin; Huang, Sijie; He, Xinheng; Wu, Kai; Zhang, Xinyue; Yang, Dehua; Xie, Xin; Xu, H Eric

Distinct structural mechanisms of LGR4 modulation by Norrin and RSPOs in Wnt/β-catenin signaling

Norrin和RSPOs在Wnt/β-catenin信号通路中对LGR4调控的不同结构机制

Qiao, Huarui; Hu, Fangzheng; Wang, Yiang; Wang, Lu; Zhou, Siyu; Guo, Shaojue; Xu, Yiwen; Xu, Jianfeng; Cui, Qianqian; Yang, Qilun; Xu, H Eric; Zhu, Jianwei; Geng, Yong

Structural insights into antagonist recognition by the vasopressin V2 receptor

血管加压素V2受体拮抗剂识别的结构解析

Zhang, Tianwei; Liu, Hongli; You, Chongzhao; Zhang, Yixiao; Xu, Youwei; Pan, Benxun; Wu, Canrong; Jin, Sanshan; Yin, Yu-Ling; Wu, Kai; Chen, Yue; Sun, Hong; Si, Yuan; Tan, Yangxia; Yin, Wanchao; Xu, H Eric; Guo, Dong; Jiang, Yi