日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Efficient Method for High-Throughput Screening of Compound Libraries Targeting Human PD-L1

高效筛选靶向人PD-L1化合物库的方法

Zamani, Mohammad Reza; Čermáková, Kateřina; Hadzima, Martin; Šácha, Pavel; Konvalinka, Jan

On-Resin Assembly of Macrocyclic Inhibitors of Cryptococcus neoformans May1: A Pathway to Potent Antifungal Agents.

新型隐球菌 May1 大环抑制剂的树脂上组装:通往强效抗真菌剂的途径

Kryštůfek Robin, Verner Václav, Šácha Pavel, Hadzima Martin, Trajhan Filip, Starková Jana, Tloušt'ová Eva, Dvořáková Alexandra, Pecina Adam, Brynda Jiří, Chalupský Karel, Hájek Miroslav, Boucher Michael J, Majer Pavel, Řezáč Jan, Madhani Hiten D, Craik Charles S, Konvalinka Jan

Uncovering the glutamate carboxypeptidase II microenvironment using a multi-labeling proteomic approach

利用多标记蛋白质组学方法揭示谷氨酸羧肽酶II的微环境

Pokorná, Jana; Hadzima, Martin; Křenková, Alena; Smith, Joshua D; Šubr, Vladimír; Kryštůfek, Robin; Hubálek, Martin; Starková, Jana; Šrámková, Karolína; Etrych, Tomáš; Kostka, Libor; Sedlák, František; Konvalinka, Jan; Šácha, Pavel

Identification of 6‑Aryl-7-Deazapurine Ribonucleoside Phosphonates as Inhibitors of Ecto-5'-Nucleotidase (CD73).

鉴定 6'芳基-7-脱氮嘌呤核糖核苷膦酸酯为外-5'-核苷酸酶 (CD73) 抑制剂

Šímová Magdalena, Ormsby Tereza, Å inkevičiuÌ tė Ugnė, Sirotová Veselovská Lucia, Čermáková Kateřina, Hadzima Martin, Bartoň Lenka, Staňurová Jana, Kramná Anežka, Šácha Pavel, Tichý Michal, Hocek Michal, Konvalinka Jan, Blazkova Kristyna

Polymer-Tethered Quenched Fluorescent Probes for Enhanced Imaging of Tumor-Associated Proteases

用于增强肿瘤相关蛋白酶成像的聚合物连接淬灭荧光探针

Hadzima, Martin; Faucher, Franco F; Blažková, Kristýna; Yim, Joshua J; Guerra, Matteo; Chen, Shiyu; Woods, Emily C; Park, Ki Wan; Šácha, Pavel; Šubr, Vladimír; Kostka, Libor; Etrych, Tomáš; Majer, Pavel; Konvalinka, Jan; Bogyo, Matthew

Polymer-tethered quenched fluorescent probes for enhanced imaging of tumor associated proteases

用于增强肿瘤相关蛋白酶成像的聚合物连接淬灭荧光探针

Hadzima, Martin; Faucher, Franco; Blažková, Kristýna; Yim, Joshua J; Guerra, Matteo; Chen, Shiyu; Woods, Emily C; Park, Ki Wan; Šácha, Pavel; Šubr, Vladimír; Kostka, Libor; Etrych, Tomáš; Majer, Pavel; Konvalinka, Jan; Bogyo, Matthew

Identification of specific carbonic anhydrase inhibitors via in situ click chemistry, phage-display and synthetic peptide libraries: comparison of the methods and structural study

利用原位点击化学、噬菌体展示和合成肽库鉴定特异性碳酸酐酶抑制剂:方法比较和结构研究

Kugler, Michael; Hadzima, Martin; Dzijak, Rastislav; Rampmaier, Robert; Srb, Pavel; Vrzal, Lukáš; Voburka, Zdeněk; Majer, Pavel; Řezáčová, Pavlína; Vrabel, Milan