日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A strategy for liver selective NRF2 induction via cytochrome P450-activated prodrugs with low activity in hypoxia.

一种通过细胞色素 P450 激活的前药诱导肝脏选择性 NRF2 的策略,该前药在缺氧条件下活性较低

Ng Mei Ying, Hagen Thilo

Conjugating uncoupler compounds with hydrophobic hydrocarbon chains to achieve adipose tissue selective drug accumulation

将解偶联化合物与疏水性烃链偶联,以实现药物在脂肪组织中的选择性蓄积。

Ng, Mei Ying; Song, Zhi Jian; Venkatesan, Gopalakrishnan; Rodriguez-Cuenca, Sergio; West, James A; Yang, Shili; Tan, Choon Hong; Ho, Paul Chi-Lui; Griffin, Julian L; Vidal-Puig, Antonio; Bassetto, Marcella; Hagen, Thilo

Structural investigations on the mitochondrial uncouplers niclosamide and FCCP

对线粒体解偶联剂尼克酰胺和FCCP的结构研究

Ng, Mei Ying; Song, Zhi Jian; Tan, Choon Hong; Bassetto, Marcella; Hagen, Thilo

Regulation of the NRF2 transcription factor by andrographolide and organic extracts from plant endophytes

穿心莲内酯和植物内生菌有机提取物对NRF2转录因子的调控

Wong, Daphne Pei Wen; Ng, Mei Ying; Leung, Jia Yu; Boh, Boon Kim; Lim, Ee Chien; Tan, Shi Hua; Lim, Shuying; Seah, Wen Hui; Hu, Christine Zhiwen; Ho, Boon Chuan; Ng, Daphne Hui Ping; Hagen, Thilo

Regulation of Cullin-RING ubiquitin ligase 1 by Spliceosome-associated protein 130 (SAP130)

剪接体相关蛋白130 (SAP130) 对 Cullin-RING 泛素连接酶1的调控

Cordero-Espinoza, Lucia; Hagen, Thilo

Oxygen versus Reactive Oxygen in the Regulation of HIF-1α: The Balance Tips

氧与活性氧在HIF-1α调控中的作用:平衡之道

Hagen, Thilo

Mechanism of cullin3 E3 ubiquitin ligase dimerization.

cullin3 E3泛素连接酶二聚化的机制

Choo Yin Yin, Hagen Thilo

Characterization of the role of COP9 signalosome in regulating cullin E3 ubiquitin ligase activity

阐明COP9信号体在调控cullin E3泛素连接酶活性中的作用

Choo, Yin Yin; Boh, Boon Kim; Lou, Jessica Jie Wei; Eng, Jolane; Leck, Yee Chin; Anders, Benjamin; Smith, Peter G; Hagen, Thilo

Compound C prevents Hypoxia-Inducible Factor-1α protein stabilization by regulating the cellular oxygen availability via interaction with Mitochondrial Complex I

化合物C通过与线粒体复合物I相互作用调节细胞氧气供应,从而阻止缺氧诱导因子-1α蛋白的稳定。

Chua, Yee Liu; Hagen, Thilo

Stabilization of hypoxia-inducible factor-1alpha protein in hypoxia occurs independently of mitochondrial reactive oxygen species production

缺氧条件下缺氧诱导因子-1α蛋白的稳定化与线粒体活性氧的产生无关。

Chua, Yee Liu; Dufour, Eric; Dassa, Emmanuel P; Rustin, Pierre; Jacobs, Howard T; Taylor, Cormac T; Hagen, Thilo