日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Translational molecular imaging and drug development in multiple sclerosis

多发性硬化症的转化分子影像和药物开发

Tay, Daniel; Ahmed, Hazem; Dawoud, Alyaa; Salam, Mohamed; Gobbi, Luca; Grether, Uwe; Edelmann, Martin R; Wittwer, Matthias B; Collin, Ludovic; Atz, Kenneth; Keaney, James; Giroud, Maude; Rossi, Alexia; Gennari, Antonio Giulio; Pagano, Gennaro; Parrot, Neil John; Barakovic, Muhamed; Rominger, Axel; Gebhard, Catherine; Ametamey, Simon M; Saindane, Amit M; Liang, Steven H; Haider, Achi

Preclinical development of [(18)F]TAAR1-2203 as a PET radioligand for imaging TAAR1 expression and receptor occupancy

[(18)F]TAAR1-2203 作为 PET 放射性配体用于 TAAR1 表达和受体占有率成像的临床前开发

Haider, Achi; Xiao, Zhiwei; Chen, Jiahui; Pfister, Stefanie K; Zhou, Xin; Li, Yinlong; Chaudhary, Ahmad; Zhao, Chunyu; Rong, Jian; Paehler, Axel; Mohr, Susanne; Norcross, Roger D; Honer, Michael; Mu, Linjing; Gobbi, Luca; Schibli, Roger; Hoener, Marius C; Liang, Steven H

Radiosynthesis and Evaluation of (18)F‑Labeled Deuterated Radioligand for Positron Emission Tomography Imaging of Cholesterol 24-Hydroxylase

合成和评价用于胆固醇24-羟化酶正电子发射断层扫描成像的(18)F标记氘代放射性配体

Li, Yinlong; Song, Zhendong; Shi, Haofeng; Zhao, Taoqian; Chen, Jiahui; Zhou, Xin; Hu, Qilong; Li, Xiaoyan; Meng, Lingxin; Song, Ruihu; Sun, Zhenkun; Li, Chongjiao; Haider, Achi; Yuan, Hongjie; Liang, Steven H

Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-dimensional optimization

通过反应预测和多维优化加速药物发现中的先导化合物转化进程

Nippa, David F; Atz, Kenneth; Stenzhorn, Yannick; Müller, Alex T; Tosstorff, Andreas; Benz, Jörg; Binch, Hayley; Bürkler, Markus; Haider, Achi; Heer, Dominik; Hochstrasser, Remo; Kramer, Christian; Reutlinger, Michael; Schneider, Petra; Shema, Thierry; Topp, Andreas; Walter, Alexander; Wittwer, Matthias B; Wolfard, Jens; Kuhn, Bernd; van der Stelt, Mario; Martin, Rainer E; Grether, Uwe; Schneider, Gisbert

Age modulates the link between stress-related neural activity and mortality

年龄调节应激相关神经活动与死亡率之间的联系

Mikail, Nidaa; Sablonier, Noemi; Gebert, Pimrapat; Glarner, Isabelle; Vinzens, Adriana; Haider, Achi; Todorov, Atanas; Bengs, Susan; Portmann, Angela; Treyer, Valerie; Wegener, Susanne; Gräni, Christoph; Pazhenkottil, Aju P; Gebhard, Caroline E; Regitz-Zagrosek, Vera; Tanner, Felix C; Kaufmann, Philipp A; Buechel, Ronny R; Rossi, Alexia; Gebhard, Catherine

Development of a novel (18)F-labeled reversible-binding radioligand for imaging monoacylglycerol lipase with positron emission tomography.

开发一种新型的(18)F标记可逆结合放射性配体,用于正电子发射断层扫描成像单酰甘油脂肪酶。

Rong Jian, Zhao Chunyu, Chaudhary Ahmad F, Ware Tim, Van Richard S, Li Yinlong, Calderon Leon Erick R, Dang Vivi, Chen Jiahui, Xiao Zhiwei, Zhou Xin, Zhang Wei, Bi Chunyang, Zhang Kuo, Patel Jimmy S, Shao Yihan, Ran Chongzhao, Collin Ludovic, Haider Achi, Cravatt Benjamin F, Liang Steven H

Age- and sex-specific differences in myocardial sympathetic tone and left ventricular remodeling following myocardial injury

心肌损伤后心肌交感神经张力和左心室重构的年龄和性别差异

Haider, Achi; Bengs, Susan; Portmann, Angela; Fröhlich, Sandro; Etter, Dominik; Maredziak, Monika; Warnock, Geoffrey I; Akhmedov, Alexander; Kozerke, Sebastian; Keller, Claudia; Montecucco, Fabrizio; Weber, Bruno; Mu, Linjing; Buechel, Ronny R; Regitz-Zagrosek, Vera; Kaufmann, Philipp A; Camici, Giovanni G; Ametamey, Simon M; Gebhard, Catherine

Development of a Novel (18)F-Labeled Radioligand for Imaging Phosphodiesterase 7 with Positron Emission Tomography

开发一种新型的(18)F标记放射性配体用于正电子发射断层扫描成像磷酸二酯酶7

Rong, Jian; Zhao, Chunyu; Chaudhary, Ahmad F; Jones, Evan; Van, Richard; Song, Zhendong; Li, Yinlong; Chen, Jiahui; Zhou, Xin; Patel, Jimmy S; Gao, Yabiao; Sun, Zhenkun; Feng, Siyan; Zhang, Zachary; Collier, Thomas L; Ran, Chongzhao; Haider, Achi; Shao, Yihan; Yuan, Hongjie; Liang, Steven H

Radiosynthesis and Preclinical Evaluation of a Carbon-11 Labeled Phosphodiesterase 7 Inhibitor for PET Neuroimaging

用于PET神经影像的碳-11标记磷酸二酯酶7抑制剂的放射合成和临床前评价

Xiao, Zhiwei; Sun, Jiyun; Fujinaga, Masayuki; Wei, Huiyi; Zhao, Chunyu; Haider, Achi; Van, Richard; Kuang, Shi; Yamasaki, Tomoteru; Zhang, Yiding; Rong, Jian; Hu, Kuan; Chen, Jiahui; Leon, Erick Calderon; Mori, Wakana; Xie, Lin; Wei, Junjie; Xu, Yi; Shao, Yihan; Zhang, Han-Ting; Xu, Ying; Ran, Chongzhao; Lloyd, Kc Kent; Wang, Lu; Zhang, Ming-Rong; Liang, Steven H

Radiosynthesis and Evaluation of (11)C‑Labeled Imidazolyl Pyrimidine Derivatives for Positron Emission Tomography Imaging of Glycogen Synthase Kinase‑3

利用放射合成和评价(11)C标记的咪唑基嘧啶衍生物对糖原合成酶激酶-3进行正电子发射断层扫描成像

Li, Yinlong; Dahl, Kenneth; Elmore, Charles S; Sandell, Johan; Takano, Akihiro; Halldin, Christer; Farde, Lars; Ahlgren, Charlotte; Cochrane, Alison; Rong, Jian; Chen, Jiahui; Zhao, Chunyu; Zhou, Xin; Patel, Jimmy S; Song, Zhendong; Chaudhary, Ahmad; Gao, Yabiao; Sun, Zhenkun; Zhang, Zachary; Feng, Siyan; Haider, Achi; Liang, Steven H; Schou, Magnus