Metabolic Activation versus Masked Prodrugs: Bisubstrate Mimic Inhibitors of CoaBC's PPCS Activity in Mycobacterium tuberculosis and Staphylococcus aureus
代谢活化与掩蔽前药:结核分枝杆菌和金黄色葡萄球菌中CoaBC PPCS活性的双底物模拟抑制剂
期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.5c00047
Kotzé, Timothy J; Mostert, Konrad J; Domingo, Riyad; Wang, Xu; Moolman, Wessel J A; Butman, Hailey S; Pepin, Abigail; McKay, Kyle T; Neveling, Deon P; Evans, Joanna C; Mizrahi, Valerie; van Otterlo, Willem A L; Dowd, Cynthia S; Strauss, Erick