日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An all-in-one pipeline for the in vitro discovery and in vivo testing of Plasmodium falciparum malaria transmission blocking drugs.

用于体外发现和体内测试恶性疟原虫疟疾传播阻断药物的一体化流程

Brancucci Nicolas M B, Gumpp Christin, van Gemert Geert-Jan, Yu Xiao, Passecker Armin, Nardella Flore, Thommen Basil T, Chambon Marc, Turcatti Gerardo, Halby Ludovic, Blasco Benjamin, Duffey Maëlle, Arimondo Paola B, Bousema Teun, Scherf Artur, Leroy Didier, Kooij Taco W A, Rottmann Matthias, Voss Till S

Design, synthesis and evaluation of pyrimidinobenzylamide and pyrimidinothiophenamide derivatives as inhibitors of DOT1L and related epigenetic targets DNMT3a, PRMT4 and other HMTs

设计、合成和评价嘧啶并苄酰胺和嘧啶并噻吩酰胺衍生物作为DOT1L及相关表观遗传靶点DNMT3a、PRMT4和其他HMTs的抑制剂

Castillo-Aguilera, Oscar Omar; Depreux, Patrick; Halby, Ludovic; Bailly, Christian; Domínguez-Ramírez, Lenin; Gul, Sheraz; Arimondo, Paola B; Goossens, Laurence

Towards the sustainable discovery and development of new antibiotics

迈向新型抗生素的可持续发现和开发

Miethke, Marcus; Pieroni, Marco; Weber, Tilmann; Brönstrup, Mark; Hammann, Peter; Halby, Ludovic; Arimondo, Paola B; Glaser, Philippe; Aigle, Bertrand; Bode, Helge B; Moreira, Rui; Li, Yanyan; Luzhetskyy, Andriy; Medema, Marnix H; Pernodet, Jean-Luc; Stadler, Marc; Tormo, José Rubén; Genilloud, Olga; Truman, Andrew W; Weissman, Kira J; Takano, Eriko; Sabatini, Stefano; Stegmann, Evi; Brötz-Oesterhelt, Heike; Wohlleben, Wolfgang; Seemann, Myriam; Empting, Martin; Hirsch, Anna K H; Loretz, Brigitta; Lehr, Claus-Michael; Titz, Alexander; Herrmann, Jennifer; Jaeger, Timo; Alt, Silke; Hesterkamp, Thomas; Winterhalter, Mathias; Schiefer, Andrea; Pfarr, Kenneth; Hoerauf, Achim; Graz, Heather; Graz, Michael; Lindvall, Mika; Ramurthy, Savithri; Karlén, Anders; van Dongen, Maarten; Petkovic, Hrvoje; Keller, Andreas; Peyrane, Frédéric; Donadio, Stefano; Fraisse, Laurent; Piddock, Laura J V; Gilbert, Ian H; Moser, Heinz E; Müller, Rolf

Direct Synthesis of Allyl Amines with 2-Nitrosulfonamide Derivatives via the Tsuji-Trost Reaction

利用辻-特罗斯特反应直接合成2-硝基磺酰胺衍生物烯丙胺

Bon, Corentin; Arimondo, Paola B; Halby, Ludovic

DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites

DNA甲基化双底物抑制剂是速效药物,可有效对抗青蒿素耐药的恶性疟原虫。

Nardella, Flore; Halby, Ludovic; Hammam, Elie; Erdmann, Diane; Cadet-Daniel, Véronique; Peronet, Roger; Ménard, Didier; Witkowski, Benoit; Mecheri, Salah; Scherf, Artur; Arimondo, Paola B

Sequence-specific targeting of IGF-I and IGF-IR genes by camptothecins

喜树碱对IGF-I和IGF-IR基因的序列特异性靶向作用

Oussedik, Kahina; François, Jean-Christophe; Halby, Ludovic; Senamaud-Beaufort, Catherine; Toutirais, Géraldine; Dallavalle, Sabrina; Pommier, Yves; Pisano, Claudio; Arimondo, Paola B

Sequence-specific DNA cleavage mediated by bipyridine polyamide conjugates

联吡啶聚酰胺缀合物介导的序列特异性DNA切割

Simon, Philippe; Cannata, Fabio; Perrouault, Loïc; Halby, Ludovic; Concordet, Jean-Paul; Boutorine, Alexandre; Ryabinin, Vladimir; Sinyakov, Alexandre; Giovannangeli, Carine

The triple helix: 50 years later, the outcome

三螺旋结构:50年后的结果

Duca, Maria; Vekhoff, Pierre; Oussedik, Kahina; Halby, Ludovic; Arimondo, Paola B

Molecular basis of the targeting of topoisomerase II-mediated DNA cleavage by VP16 derivatives conjugated to triplex-forming oligonucleotides

VP16衍生物与三链形成寡核苷酸偶联后靶向拓扑异构酶II介导的DNA切割的分子基础

Duca, Maria; Guianvarc'h, Dominique; Oussedik, Kahina; Halby, Ludovic; Garbesi, Anna; Dauzonne, Daniel; Monneret, Claude; Osheroff, Neil; Giovannangeli, Carine; Arimondo, Paola B

Exploring the cellular activity of camptothecin-triple-helix-forming oligonucleotide conjugates

探索喜树碱-三螺旋形成寡核苷酸缀合物的细胞活性

Arimondo, Paola B; Thomas, Craig J; Oussedik, Kahina; Baldeyrou, Brigitte; Mahieu, Christine; Halby, Ludovic; Guianvarc'h, Dominique; Lansiaux, Amélie; Hecht, Sidney M; Bailly, Christian; Giovannangeli, Carine