日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploring Alternative Zinc-Binding Groups in Histone Deacetylase (HDAC) Inhibitors Uncovers DS-103 as a Potent Ethylhydrazide-Based HDAC Inhibitor with Chemosensitizing Properties.

探索组蛋白去乙酰化酶 (HDAC) 抑制剂中的替代锌结合基团,发现 DS-103 是一种具有化学增敏特性的强效乙基肼基 HDAC 抑制剂

Stopper Daniel, Biermann Lukas, Watson Paris R, Li Jingyu, König Beate, Gaynes Matthew N, Pessanha de Carvalho Lais, Klose Jana, Hanl Maria, Hamacher Alexandra, Schäker-Hübner Linda, Ramsbeck Daniel, Held Jana, Christianson David W, Kassack Matthias U, Hansen Finn K

Oxa Analogues of Nexturastat A Demonstrate Improved HDAC6 Selectivity and Superior Antileukaemia Activity

Nexturastat A 的氧杂类似物表现出更高的 HDAC6 选择性和更优异的抗白血病活性

Pflieger, Marc; Sönnichsen, Melf; Horstick-Muche, Nadine; Yang, Jing; Schliehe-Diecks, Julian; Schöler, Andrea; Borkhardt, Arndt; Hamacher, Alexandra; Kassack, Matthias U; Hansen, Finn K; Bhatia, Sanil; Kurz, Thomas

Hydroxamic Acids Immobilized on Resins (HAIRs): Synthesis of Dual-Targeting HDAC Inhibitors and HDAC Degraders (PROTACs)

树脂上固定的羟肟酸(HAIRs):双靶向HDAC抑制剂和HDAC降解剂(PROTACs)的合成

Sinatra, Laura; Bandolik, Jan J; Roatsch, Martin; Sönnichsen, Melf; Schoeder, Clara T; Hamacher, Alexandra; Schöler, Andrea; Borkhardt, Arndt; Meiler, Jens; Bhatia, Sanil; Kassack, Matthias U; Hansen, Finn K

Multicomponent Synthesis and Binding Mode of Imidazo[1,2- a]pyridine-Capped Selective HDAC6 Inhibitors

咪唑并[1,2-a]吡啶封端的选择性HDAC6抑制剂的多组分合成及结合模式

Mackwitz, Marcel K W; Hamacher, Alexandra; Osko, Jeremy D; Held, Jana; Schöler, Andrea; Christianson, David W; Kassack, Matthias U; Hansen, Finn K

Structure-Activity Study of Dihydrocinnamic Acids and Discovery of the Potent FFA1 (GPR40) Agonist TUG-469

二氢肉桂酸的结构活性研究及强效FFA1(GPR40)激动剂TUG-469的发现

Christiansen, Elisabeth; Due-Hansen, Maria E; Urban, Christian; Merten, Nicole; Pfleiderer, Michael; Karlsen, Kasper K; Rasmussen, Sanne S; Steensgaard, Mette; Hamacher, Alexandra; Schmidt, Johannes; Drewke, Christel; Petersen, Rasmus Koefoed; Kristiansen, Karsten; Ullrich, Susanne; Kostenis, Evi; Kassack, Matthias U; Ulven, Trond