日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and optimization of simplified inhibitors targeting Escherichia coli and Klebsiella pneumoniae IspE

设计和优化针对大肠杆菌和肺炎克雷伯菌 IspE 的简化抑制剂

Walsh, Danica J; Hamid, Rawia; Giele, Tim; Reiling, Norbert; Rottmann, Matthias; Hamed, Mostafa M; Hirsch, Anna K H

Fragment Discovery by X-Ray Crystallographic Screening Targeting the CTP Binding Site of Pseudomonas Aeruginosa IspD

利用X射线晶体学筛选发现靶向铜绿假单胞菌IspD CTP结合位点的片段

Willocx, Daan; D'Auria, Lucia; Walsh, Danica; Scherer, Hugo; Alhayek, Alaa; Hamed, Mostafa M; Borel, Franck; Diamanti, Eleonora; Hirsch, Anna K H

A Novel Antimalarial Agent that Inhibits Protein Synthesis in Plasmodium falciparum

一种新型抗疟药,可抑制恶性疟原虫的蛋白质合成

Bravo, Patricia; Diamanti, Eleonora; Hamed, Mostafa M; Bizzarri, Lorenzo; Wiedemar, Natalie; Passecker, Armin; Brancucci, Nicolas M B; Albisetti, Anna; Gumpp, Christin; Illarionov, Boris; Fischer, Markus; Witschel, Matthias; Schehl, Tobias; Hahne, Hannes; Mäser, Pascal; Rottmann, Matthias; Hirsch, Anna K H

Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity

抗疟化合物中的正电荷可释放广谱抗菌活性

Braun-Cornejo, Maria; Platteschorre, Mitchell; de Vries, Vincent; Bravo, Patricia; Sonawane, Vidhisha; Hamed, Mostafa M; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K H

Nanoparticles in liposomes: a platform for increased antibiotic selectivity in multidrug resistant bacteria in respiratory tract infections.

脂质体中的纳米颗粒:提高呼吸道感染中多重耐药菌抗生素选择性的平台

Fakhoury Nathalie E, Mansour Samar, Abdel-Halim Mohammad, Hamed Mostafa M, Empting Martin, Boese Annette, Loretz Brigitta, Lehr Claus-Michael, Tammam Salma N

Fragment Based Drug Discovery by Microscale Thermophoresis Targeting Klebsiella pneumoniae and Escherichia coli IspE

基于微尺度热泳的片段药物发现靶向肺炎克雷伯菌和大肠杆菌IspE

Walsh, Danica J; Willocx, Daan; Hamid, Rawia; Hamed, Mostafa M; Hirsch, Anna K H

Targeting the Plasmodium falciparum IspE Enzyme

靶向恶性疟原虫 IspE 酶

Diamanti, Eleonora; Steinbach, Annina M; de Carvalho, Lais P; Ropponen, Henni-Karoliina; Lacour, Antoine; Hamid, Rawia; Eisa, Sidra; Bravo, Patricia; Bousis, Spyridon; Illarionov, Boris; Fischer, Markus; Hamed, Mostafa M; Bach, Nina C; Rottmann, Matthias; Held, Jana; Witschel, Matthias; Sieber, Stephan A; Hirsch, Anna K H

Characterization, modeling, and anticancer activity of L.arginase production from marine Bacillus licheniformis OF2

海洋地衣芽孢杆菌 OF2 产生的 L.精氨酸酶的表征、建模和抗癌活性

Manal S Selim, Marwa M Mounier, Sayeda A Abdelhamid, Ahmed Abdelghani Hamed, Mostafa M Abo Elsoud, Sahar S Mohamed

Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof-of-Principle

PqsR反向激动剂转化研究进展:从体外功效优化到体内原理验证

Hamed, Mostafa M; Abdelsamie, Ahmed S; Rox, Katharina; Schütz, Christian; Kany, Andreas M; Röhrig, Teresa; Schmelz, Stefan; Blankenfeldt, Wulf; Arce-Rodriguez, Alejandro; Borrero-de Acuña, José Manuel; Jahn, Dieter; Rademacher, Jessica; Ringshausen, Felix C; Cramer, Nina; Tümmler, Burkhard; Hirsch, Anna K H; Hartmann, Rolf W; Empting, Martin

Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters

结构导向的小分子叶酸摄取抑制剂优化:靶向能量耦合因子转运蛋白

Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hirsch, Anna K H