日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural and Biophysical Analyses of Human Prostamide/Prostaglandin F Synthase with Two Active Form-Mimicking Mutations

人前列腺素/前列腺素F合成酶两种活性模拟突变体的结构和生物物理分析

Cheon, Sang Won; Nguyen, Yen Thi Kim; Kang, Jin Mo; Yu, Youngbeom; Heo, Yoonyoung; Kim, Hyoun Sook; Han, Byung Woo

Impaired chaperone-mediated autophagy leads to abnormal SORT1 (sortilin 1) turnover and CES1-dependent triglyceride hydrolysis.

分子伴侣介导的自噬受损会导致 SORT1(sortilin 1)周转异常和 CES1 依赖性甘油三酯水解

Choi You-Jin, Nam Yoon Ah, Hyun Ji Ye, Yu Jihyeon, Mun Yewon, Yun Sung Ho, Lee Wonseok, Park Cheon Jun, Han Byung Woo, Lee Byung-Hoon

Design, Synthesis, and Biological Evaluation of 5',7-Disubstituted 7-Deaza-adenosine Analogues as Irreversible Pan-FGFR Inhibitors

5',7-二取代7-脱氮腺苷类似物作为不可逆泛FGFR抑制剂的设计、合成和生物学评价

Park, Jung Hoon; Tran, Phuong Thao; Ko, Hye Lin; Mun, Seonghee; Jang, Sung Chul; Moon, Dong Hyun; Han, Jaeho; Kim, Jieun; Kim, Gibae; Choi, Hongseok; Kim, Seung Woo; Kim, Minjae; Lee, Sang Kook; Han, Byung Woo; Kang, Keon Wook; Jeong, Lak Shin

Martinostat as a novel HDAC inhibitor to overcome tyrosine kinase inhibitor resistance in chronic myeloid leukemia.

Martinostat 是一种新型 HDAC 抑制剂,可克服慢性粒细胞白血病中的酪氨酸激酶抑制剂耐药性

Yang Haeun, Li Vladimir, Park Su Jung, Cheon Sang Won, Lorant Anne, Mazumder Aloran, Lee Jin Young, Orlikova-Boyer Barbora, Cerella Claudia, Christov Christo, Kirsch Gilbert, Olberg Dag Erlend, Bormans Guy, Kang Hyoung Jin, Han Byung Woo, Schnekenburger Michael, Diederich Marc

Structural insight into the distinct regulatory mechanism of the HEPN-MNT toxin-antitoxin system in Legionella pneumophila

军团菌中 HEPN-MNT 毒素-抗毒素系统独特调控机制的结构解析

Jin, Chenglong; Jeon, Cha-Hee; Kim, Heung Wan; Kang, Jin Mo; Choi, Yuri; Kang, Sung-Min; Lee, Hyung Ho; Kim, Do-Hee; Han, Byung Woo; Lee, Bong-Jin

ATP1A1/BCL2L1 predicts the response of myelomonocytic and monocytic acute myeloid leukemia to cardiac glycosides

ATP1A1/BCL2L1 可预测髓单核细胞性急性髓系白血病和单核细胞性急性髓系白血病对强心苷的反应。

Cerella, Claudia; Gajulapalli, Sruthi Reddy; Lorant, Anne; Gerard, Deborah; Muller, Florian; Lee, Yejin; Kim, Kyung Rok; Han, Byung Woo; Christov, Christo; Récher, Christian; Sarry, Jean-Emmanuel; Dicato, Mario; Diederich, Marc

In Silico Discovery of 5'-Modified 7-Deoxy-7-ethynyl-4'-thioadenosine as a HASPIN Inhibitor and Its Synergistic Anticancer Effect with the PLK1 Inhibitor

利用计算机模拟发现 5'-修饰的 7-脱氧-7-乙炔基-4'-硫代腺苷作为 HASPIN 抑制剂及其与 PLK1 抑制剂的协同抗癌作用

Kwon, Eun-Ji; Mashelkar, Karishma K; Seo, Juhee; Shin, Yoon-Ze; Sung, Kisu; Jang, Sung Chul; Cheon, Sang Won; Lee, Haeseung; Lee, Hyuk Woo; Kim, Gyudong; Han, Byung Woo; Lee, Sang Kook; Jeong, Lak Shin; Cha, Hyuk-Jin

In Memoriam: Seung Ki Lee (1944-2022)

悼念:李升基(1944-2022)

Carroll, Dana; Surh, Young-Joon; Lee, Jung-Weon; Diederich, Marc; Han, Byung Woo; Cha, Hyuk-Jin; Kim, Kyu-Won

Reaction hijacking inhibition of Plasmodium falciparum asparagine tRNA synthetase

恶性疟原虫天冬酰胺tRNA合成酶的反应劫持抑制

Xie, Stanley C; Wang, Yinuo; Morton, Craig J; Metcalfe, Riley D; Dogovski, Con; Pasaje, Charisse Flerida A; Dunn, Elyse; Luth, Madeline R; Kumpornsin, Krittikorn; Istvan, Eva S; Park, Joon Sung; Fairhurst, Kate J; Ketprasit, Nutpakal; Yeo, Tomas; Yildirim, Okan; Bhebhe, Mathamsanqa N; Klug, Dana M; Rutledge, Peter J; Godoy, Luiz C; Dey, Sumanta; De Souza, Mariana Laureano; Siqueira-Neto, Jair L; Du, Yawei; Puhalovich, Tanya; Amini, Mona; Shami, Gerry; Loesbanluechai, Duangkamon; Nie, Shuai; Williamson, Nicholas; Jana, Gouranga P; Maity, Bikash C; Thomson, Patrick; Foley, Thomas; Tan, Derek S; Niles, Jacquin C; Han, Byung Woo; Goldberg, Daniel E; Burrows, Jeremy; Fidock, David A; Lee, Marcus C S; Winzeler, Elizabeth A; Griffin, Michael D W; Todd, Matthew H; Tilley, Leann

Structural basis for SdgB- and SdgA-mediated glycosylation of staphylococcal adhesive proteins

葡萄球菌黏附蛋白SdgB和SdgA介导的糖基化的结构基础

Kim, Dong Gyun; Baek, Inwha; Lee, Yeon; Kim, Hyerry; Kim, Jin Young; Bang, Geul; Kim, Sunghwan; Yoon, Hye Jin; Han, Byung Woo; Suh, Se Won; Kim, Hyoun Sook