日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The primary mechanism for highly potent inhibition of HIV-1 maturation by lenacapavir.

lenacapavir 高效抑制 HIV-1 成熟的主要机制

Huang Szu-Wei, Briganti Lorenzo, Annamalai Arun S, Greenwood Juliet, Shkriabai Nikoloz, Haney Reed, Armstrong Michael L, Wempe Michael F, Singh Satya Prakash, Francis Ashwanth C, Engelman Alan N, Kvaratskhelia Mamuka

Erratum for Dinh et al., "The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir"

更正:Dinh 等人,“病毒对变构 HIV-1 整合酶抑制剂 pirmitegravir 产生耐药性的结构和机制基础”

Dinh, Tung; Tber, Zahira; Rey, Juan S; Mengshetti, Seema; Annamalai, Arun S; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F; Perilla, Juan R; Kim, Baek; Kvaratskhelia, Mamuka

Structural and mechanistic bases for resistance of the M66I capsid variant to lenacapavir.

M66I衣壳变体对lenacapavir产生耐药性的结构和机制基础

Briganti Lorenzo, Annamalai Arun S, Bester Stephanie M, Wei Guochao, Andino-Moncada Jonathan R, Singh Satya P, Kleinpeter Alex B, Tripathi Meghna, Nguyen Binh, Radhakrishnan Rajalingam, Singh Parmit K, Greenwood Juliet, Schope Lauren I, Haney Reed, Huang Szu-Wei, Freed Eric O, Engelman Alan N, Francis Ashwanth C, Kvaratskhelia Mamuka

Delineating Structural Functionalities of Lenacapavir Amenable to Modifications for Targeting Emerging Drug-Resistant HIV‑1 Capsid Variants

阐明利那卡帕韦的结构功能,以便对其进行修饰,从而靶向新出现的耐药性 HIV-1 衣壳变体

Adu-Ampratwum, Daniel; Annamalai, Arun S; Dinh, Tung; Lockwood, Jeffrey R; Bockbrader, Ross H; Haney, Reed; Kvaratskhelia, Mamuka; Fuchs, James R

The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir

病毒对变构HIV-1整合酶抑制剂吡米特格拉韦产生耐药性的结构和机制基础

Dinh, Tung; Tber, Zahira; Rey, Juan S; Mengshetti, Seema; Annamalai, Arun S; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F; Perilla, Juan R; Kim, Baek; Kvaratskhelia, Mamuka

Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions

喹啉酮衍生物作为HIV-1整合酶催化位点和整合酶-RNA相互作用的双重抑制剂

Patacchini, Elisa; Madia, Valentina Noemi; Albano, Aurora; Ruggieri, Giuseppe; Messore, Antonella; Ialongo, Davide; Saccoliti, Francesco; Scipione, Luigi; Cosconati, Sandro; Koneru, Pratibha C; Haney, Reed; Kvaratskhelia, Mamuka; Di Santo, Roberto; Costi, Roberta