日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

Correction: Bortezomib-releasing silica-collagen xerogels for local treatment of osteolytic bone- and minimal residual disease in multiple myeloma

更正:用于局部治疗多发性骨髓瘤溶骨性骨病和微小残留病灶的硼替佐米释放二氧化硅-胶原蛋白干凝胶

Hose, Dirk; Ray, Seemun; Rößler, Sina; Thormann, Ulrich; Schnettler, Reinhard; de Veirman, Kim; Khassawna, Thaqif El; Heiss, Christian; Hild, Anne; Zahner, Daniel; Alagboso, Francisca; Henss, Anja; Beck, Susanne; Emde-Rajaratnam, Martina; Burhenne, Jürgen; Bamberger, Juliane; Menu, Eline; de Bruyne, Elke; Gelinsky, Michael; Kampschulte, Marian; Rohnke, Marcus; Wenisch, Sabine; Vanderkerken, Karin; Hanke, Thomas; Seckinger, Anja; Alt, Volker

Crystallographic fragment screening reveals ligand hotspots in TRIM21 PRY-SPRY domain.

晶体学片段筛选揭示了TRIM21 PRY-SPRY结构域中的配体热点

Kim Yeojin, Lučić Aleksandar, Lenz Christopher, Farges Frederic, Schwalm Martin P, Saxena Krishna, Hanke Thomas, Marples Peter G, Aschenbrenner Jasmin C, Fearon Daren, von Delft Frank, Krämer Andreas, Knapp Stefan

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

BDNF improves the survival of mesenchymal stem cells cultured on pre-structured gelatin material containing strontium and calcium phosphates for bone regeneration

BDNF可提高在含有锶和磷酸钙的预结构化明胶材料上培养的间充质干细胞的存活率,从而促进骨再生。

Itting, Paul T; Kruppke, Benjamin; Hanke, Thomas; Vijayan, Vinu; Heiss, Christian; Lips, Katrin Susanne

Un-LOK-ing a New Approach for Conformational Selective Targeting of STK10 (LOK)

针对 STK10 (LOK) 构象选择性靶向的新方法——解构 LOK

Dettenhöfer, Martina; Tandara, Laura Nadine; Amrhein, Jennifer Alisa; Kurz, Christian Georg; Schwalm, Martin Peter; Mensing, Theresa Elisabeth; Wahl, Laurenz Maximilian; Krämer, Andreas; Gerninghaus, Joshua; Lenz, Christopher; Elson, Lewis; Berger, Benedict-Tilman; Schröder, Martin; Saxena, Krishna; Müller, Susanne; Knapp, Stefan; Greco, Francesco Aleksy; Hanke, Thomas

Repurposing of the RIPK1-Selective Benzo[1,4]oxazepin-4-one Scaffold for the Development of a Type III LIMK1/2 Inhibitor.

RIPK1 选择性苯并[1,4]氧氮杂环庚酮-4-酮骨架的再利用,用于开发 III 型 LIMK1/2 抑制剂

Mandel Sebastian, Hanke Thomas, Mathea Sebastian, Chatterjee Deep, Saraswati Hayuningbudi, Berger Benedict-Tilman, Schwalm Martin Peter, Yamamoto Satoshi, Tawada Michiko, Takagi Terufumi, Ahmed Mahmood, Röhm Sandra, Corrionero Ana, Alfonso Patricia, Baena Maria, Elson Lewis, Menge Amelie, Krämer Andreas, Pereira Raquel, Müller Susanne, Krause Daniela S, Knapp Stefan

Back-Pocket Optimization of 2-Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors.

2-氨基嘧啶基大环化合物的后口袋优化可得到强效的EPHA2/GAK激酶抑制剂

Gerninghaus Joshua, Zhubi Rezart, Krämer Andreas, Karim Marwah, Tran Do Hoang Nhu, Joerger Andreas C, Schreiber Christian, Berger Lena M, Berger Benedict-Tilman, Ehret Theresa A L, Elson Lewis, Lenz Christopher, Saxena Krishna, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

How to Get Them off?-Assessment of Innovative Techniques for Generation and Detachment of Mature Osteoclasts for Biomaterial Resorption Studies

如何去除它们?——用于生物材料吸收研究的成熟破骨细胞生成和脱落的创新技术评估

Heinemann, Christiane; Adam, Josephine; Kruppke, Benjamin; Hintze, Vera; Wiesmann, Hans-Peter; Hanke, Thomas

3D Plotting of Silica/Collagen Xerogel Granules in an Alginate Matrix for Tissue-Engineered Bone Implants

用于组织工程骨植入物的藻酸盐基质中二氧化硅/胶原蛋白干凝胶颗粒的三维绘图

Rößler, Sina; Brückner, Andreas; Kruppke, Iris; Wiesmann, Hans-Peter; Hanke, Thomas; Kruppke, Benjamin