PROTAC-Mediated Degradation of Bruton's Tyrosine Kinase Is Inhibited by Covalent Binding
PROTAC 介导的布鲁顿酪氨酸激酶降解被共价结合抑制
期刊:ACS Chemical Biology
影响因子:3.5
doi:10.1021/acschembio.8b01094
Christopher P Tinworth, Hannah Lithgow, Lars Dittus, Zuni I Bassi, Sophie E Hughes, Marcel Muelbaier, Han Dai, Ian E D Smith, William J Kerr, Glenn A Burley, Marcus Bantscheff, John D Harling