日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: GluN2A-NMDA receptor inhibition disinhibits the prefrontal cortex, reduces forced swim immobility, and impairs sensorimotor gating

更正:GluN2A-NMDA受体抑制可解除前额叶皮层的抑制,减少强迫游泳引起的静止不动,并损害感觉运动门控。

Dong, Yuan-Ping; Wu, Yun; Zhao, Yi-Lu; Chen, Yu-Min; Liu, Tong-Ye; Zhang, Yi-He; Xie, Jie-Ying; Zhang, Jin-Feng; Zhang, Han; Chen, He; Peng, Yu; Zhang, Chun-Lei; Rau, Andrew R; Hansen, Kasper B; Xu, Hai-Bing; Yi, Feng

UCM-A86 is a selective positive allosteric modulator of GluN1/GluN3 NMDA receptors

UCM-A86 是 GluN1/GluN3 NMDA 受体的选择性正向变构调节剂。

Benton, Avery J; Johns, Mia R; Diamant, Emil; Rouzbeh, Nirvan; Sørensen, Valdemar P; Anderson, Carly M; Secci, Davide; Zhang, Zhucheng; Rau, Andrew R; Clausen, Rasmus P; Hansen, Kasper B

Novel binding mode for negative allosteric NMDA receptor modulators

负变构NMDA受体调节剂的新型结合模式

Lotti, James S; Syrenne, Jed T; Benton, Avery J; Al-Mousawi, Ahmad; Cornelison, Lauren E; Trolinder, Christopher J; Yi, Feng; Zhang, Zhucheng; Yates-Hansen, Cindee K; McClelland, Levi J; Bosco, James; Rau, Andrew R; Clausen, Rasmus P; Hansen, Kasper B

Native architecture, allosteric modulation and gating mechanism of glycine-dependent NMDA receptors

甘氨酸依赖性NMDA受体的天然结构、变构调节和门控机制

Kim, Junhoe; Benton, Avery J; Lotti, James S; Rouzbeh, Nirvan; Hansen, Kasper B; Gouaux, Eric

A galactose-based auto-expression system improves T7-inducible protein production in Escherichia coli.

基于半乳糖的自表达系统可提高大肠杆菌中 T7 诱导蛋白的产量

Bosco James, Gagliano Emily, Boshae Kassandra L, Statz John P, Wheeler Timothy B, Cuello DeAnna, Sliter Ashlyn, Newby Christian, Lin Bernice, Demeler Aysha, Pierpont C Logan, Yates-Hansen Cindee, Sydor Matthew J, Ferrini Maria E, Kuch Kellie C, Cooper Brandon S, Piggott Beverly J, Certel Sarah J, Hansen Kasper B, Sprang Stephen R, Bowler Bruce, McClelland Levi, Berkmen Mehmet, Voronina Ekaterina

Evaluation of allosteric N-methyl-d-aspartate receptor modulation by GluN2A-selective antagonists using pharmacological equilibrium modeling

利用药理平衡模型评估GluN2A选择性拮抗剂对N-甲基-D-天冬氨酸受体的变构调节作用

Lotti, James S; Jones, Jaron; Farnsworth, Jill C; Yi, Feng; Zhao, Fabao; Menniti, Frank S; Volkmann, Robert A; Clausen, Rasmus P; Hansen, Kasper B

UCM-A86 is a selective positive allosteric modulator of GluN1/GluN3 NMDA receptors

UCM-A86 是 GluN1/GluN3 NMDA 受体的选择性正向变构调节剂。

Benton, Avery J; Johns, Mia R; Diamant, Emil; Rouzbeh, Nirvan; Sørensen, Valdemar P; Anderson, Carly M; Secci, Davide; Zhang, Zhucheng; Rau, Andrew R; Clausen, Rasmus P; Hansen, Kasper B

Allosteric modulation of GluN1/GluN3 NMDA receptors by GluN1-selective competitive antagonists

GluN1选择性竞争性拮抗剂对GluN1/GluN3 NMDA受体的变构调节

Rouzbeh, Nirvan; Rau, Andrew R; Benton, Avery J; Yi, Feng; Anderson, Carly M; Johns, Mia R; Jensen, Loren; Lotti, James S; Holley, David C; Hansen, Kasper B

In vitro ADME characterization of a very potent 3-acylamino-2-aminopropionic acid-derived GluN2C-NMDA receptor agonist and its ester prodrugs

体外 ADME 表征一种高效的 3-酰氨基-2-氨基丙酸衍生的 GluN2C-NMDA 受体激动剂及其酯类前药

Bechthold, Elena; Grey, Lucie; Diamant, Emil; Schmidt, Judith; Steigerwald, Ruben; Zhao, Fabao; Hansen, Kasper B; Bunch, Lennart; Clausen, Rasmus P; Wünsch, Bernhard

Discovery of (R)-2-amino-3-triazolpropanoic acid derivatives as NMDA receptor glycine site agonists with GluN2 subunit-specific activity

发现(R)-2-氨基-3-三唑丙酸衍生物作为NMDA受体甘氨酸位点激动剂,具有GluN2亚基特异性活性

Zhao, Fabao; Mazis, Georgios; Yi, Feng; Lotti, James S; Layeux, Michael S; Schultz, Eric P; Bunch, Lennart; Hansen, Kasper B; Clausen, Rasmus P