日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Coronavirus Main Protease Inhibitors with Enhanced Brain Exposure and Potent Oral Efficacy in SARS-CoV-2 and MERS Infection Models

在SARS-CoV-2和MERS感染模型中发现具有增强脑暴露和强效口服疗效的冠状病毒主要蛋白酶抑制剂

Lizzadro, Luca; Li, Jiapeng; Taha, Taha Y; Degotte, Gilles; Detomasi, Tyler C; Zapatero-Belinchon, Francisco J; Hantz, Eric R; Huang, Sijie; Matsui, Yusuke; Henderson, Will R; McCann, Jack T; Montano, Mauricio; Rosecrans, Julia; Torres Pomares, Daniel F; McGovern, Briana L; Diaz-Tapia, Randy; Benjamin, Jared; Gordon, Mary E; Suazo, Isidora D; Settineri, Nicholas S; Diallo, Amy; Krogan, Nevan J; Shoichet, Brian K; Verba, Kliment A; Albrecht, Randy; García-Sastre, Adolfo; White, Kris M; Ott, Melanie; Craik, Charles S; Renslo, Adam R

Clinical Phenotypes of Critically Ill Patients with COVID-19 Infected with Omicron: A Nationwide Prospective Cohort Study

感染奥密克隆病毒的COVID-19重症患者的临床表型:一项全国性前瞻性队列研究

Audureau, Etienne; Bay, Pierre; Préau, Sébastien; Favory, Raphaël; Guigon, Aurélie; Heming, Nicholas; Gault, Elyanne; Pham, Tài; Chaghouri, Amal; Turpin, Matthieu; Morand-Joubert, Laurence; Jochmans, Sébastien; Pitsch, Aurélia; Meireles, Sylvie; Contou, Damien; Henry, Amandine; Roux, Damien; Le Hingrat, Quentin; Kimmoun, Antoine; Hartard, Cédric; Pène, Frédéric; L'Honneur, Anne-Sophie; Guillon, Antoine; Handala, Lynda; Tamion, Fabienne; Moisan, Alice; Daix, Thomas; Hantz, Sébastien; Delamaire, Flora; Thibault, Vincent; Darreau, Cédric; Thomin, Jean; Pawlotsky, Jean-Michel; Fourati, Slim; de Prost, Nicolas

Structure-Based Design of Reversible, Quinoline-2(1H)‑one Inhibitors of Serine- and Metallo-Carbapenemases

基于结构的可逆喹啉-2(1H)-酮类丝氨酸和金属碳青霉烯酶抑制剂的设计

Jacobs, Lian M C; Jaishankar, Priyadarshini; Zheng, Jeffrey; Hantz, Eric R; Lee, Isabel; Narramneni, Krishna; Poore, Nicholas; Torres, Nathanial; Jackson, Jessica K; Williams, Oriana; Darch, Sophie E; Shaw, Lindsey N; Chen, Yu; Renslo, Adam R

Carcinogenicity of hepatitis D virus, human cytomegalovirus, and Merkel cell polyomavirus

丁型肝炎病毒、人巨细胞病毒和默克尔细胞多瘤病毒的致癌性

Karagas, Margaret R; Kaldor, John; Michaelis, Martin; Muchengeti, Mazvita M; Alfaiate, Dulce; Argirion, Ilona; Chen, Xiaohua; Cunha, Celso; Hantz, Sébastien; Koljonen, Virve; Laude, Hélène C; Lui, Weng-Onn; Nevels, Michael M; O'Brien, Thomas R; Scheurer, Michael E; Touze, Antoine; Wiemels, Joseph L; Benbrahim-Tallaa, Lamia; de Conti, Aline; Facchin, Caterina; Madia, Federica; Pasqual, Elisa; Wedekind, Roland; Aguilera-Buenosvinos, Inmaculada; Clifford, Gary; Deng, Xiaobei; Dongoran, Rachmad A; Ezzemni, Sarra; Huang, Yue; Suonio, Eero; Zhai, Yue; Mattock, Heidi; Schubauer-Berigan, Mary K; Kunzmann, Andrew T

Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus MPro inhibitors with potent in vivo efficacy

基于结构的、具有高效体内疗效的高生物利用度、共价、广谱冠状病毒MPro抑制剂的发现

Tyler C Detomasi ,Gilles Degotte ,Sijie Huang ,Rahul K Suryawanshi ,Amy Diallo ,Luca Lizzadro ,Francisco J Zapatero-Belinchón ,Taha Y Taha ,Jiapeng Li ,Alicia L Richards ,Eric R Hantz ,Zain Alam ,Mauricio Montano ,Maria McCavitt-Malvido ,Rajesh Gumpena ,James R Partridge ,Galen J Correy ,Yusuke Matsui ,Annemarie F Charvat ,Isabella S Glenn ,Julia Rosecrans ,Jezrael L Revalde ,Dashiell Anderson ,Judd F Hultquist ,Michelle R Arkin ,R Jeffrey Neitz ,Danielle L Swaney ,Nevan J Krogan ,Brian K Shoichet ,Kliment A Verba ,Melanie Ott ,Adam R Renslo ,Charles S Craik

Long-range PCRs and next-generation sequencing to detect cytomegalovirus drug resistance-associated mutations

利用长片段PCR和新一代测序技术检测巨细胞病毒耐药相关突变

Andreani, Julien; Truffot, Aurélie; Tilloy, Valentin; Jardin, Hugo; Lespinasse, Matilda; Usal, Marie; Larrat, Sylvie; Morand, Patrice; Lupo, Julien; Hantz, Sébastien; Alain, Sophie; Germi, Raphaële

Key domains involved in the interaction and assembly of the HCMV terminase complex

参与HCMV末端酶复合物相互作用和组装的关键结构域

Gourin, C; Lefèvre, C; Flores, T; Couvreux, A; Alain, S; Ligat, G; Hantz, S

Functional and structural insights into HCMV terminase accessory proteins pUL77 and pUL93.

对 HCMV 末端酶辅助蛋白 pUL77 和 pUL93 的功能和结构进行了深入研究。

Gourin C, Di Meo F, Delmon C, Alain S, Hantz S

Targeting Human Cytomegalovirus as a Novel Approach for Glioblastoma Treatment

以人巨细胞病毒为靶点治疗胶质母细胞瘤的新方法

Flores, Thelma; Delpierre, Eloïse; Male, Ghislain; Gourin, Claire; Hantz, Sébastien; Damour, Alexia; Ligat, Gaëtan

Discovery of AVI-6451, a Potent and Selective Inhibitor of the SARS-CoV-2 ADP-Ribosylhydrolase Mac1 with Oral Efficacy in vivo

发现 AVI-6451,一种强效且选择性的 SARS-CoV-2 ADP-核糖水解酶 Mac1 抑制剂,具有口服体内疗效。

Jaishankar, Priyadarshini; Correy, Galen J; Matsui, Yusuke; Togo, Takaya; Rachman, Moira M; Stevens, Maisie G V; Hantz, Eric R; Zheng, Jeffrey; Diolaiti, Morgan E; Montano, Mauricio; Taha, Taha Y; Rosecrans, Julia; Pampel, Julius; Krogan, Nevan J; Shoichet, Brian K; Ashworth, Alan; Ott, Melanie; Fraser, James S; Renslo, Adam R