日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Probing Mercaptobenzamides as HIV Inactivators via Nucleocapsid Protein 7

通过核衣壳蛋白7探究巯基苯甲酰胺作为HIV灭活剂的作用

Saha, Mrinmoy; Scerba, Michael T; Shank, Nathaniel I; Hartman, Tracy L; Buchholz, Caitlin A; Buckheit, Robert W Jr; Durell, Stewart R; Appella, Daniel H

An analog of camptothecin inactive against Topoisomerase I is broadly neutralizing of HIV-1 through inhibition of Vif-dependent APOBEC3G degradation

一种对拓扑异构酶I无活性的喜树碱类似物,可通过抑制Vif依赖的APOBEC3G降解,广泛中和HIV-1病毒。

Bennett, Ryan P; Stewart, Ryan A; Hogan, Priscilla A; Ptak, Roger G; Mankowski, Marie K; Hartman, Tracy L; Buckheit, Robert W Jr; Snyder, Beth A; Salter, Jason D; Morales, Guillermo A; Smith, Harold C

Development of hexadecyloxypropyl tenofovir (CMX157) for treatment of infection caused by wild-type and nucleoside/nucleotide-resistant HIV.

十六烷氧基丙基替诺福韦(CMX157)的开发用于治疗由野生型和核苷/核苷酸耐药性 HIV 引起的感染

Lanier E Randall, Ptak Roger G, Lampert Bernhard M, Keilholz Laurie, Hartman Tracy, Buckheit Robert W Jr, Mankowski Marie K, Osterling Mark C, Almond Merrick R, Painter George R

Multivalent binding oligomers inhibit HIV Tat-TAR interaction critical for viral replication

多价结合寡聚体抑制HIV Tat-TAR相互作用,而这种相互作用对病毒复制至关重要。

Wang, Deyun; Iera, Jaclyn; Baker, Heather; Hogan, Priscilla; Ptak, Roger; Yang, Lu; Hartman, Tracy; Buckheit, Robert W Jr; Desjardins, Alexandre; Yang, Ao; Legault, Pascale; Yedavalli, Venkat; Jeang, Kuan-Teh; Appella, Daniel H

Inhibition of tubulin polymerization by select alkenyldiarylmethanes

某些烯基二芳基甲烷对微管蛋白聚合的抑制作用

Cullen, Matthew D; Sarkar, Taradas; Hamel, Ernest; Hartman, Tracy L; Watson, Karen M; Buckheit, Robert W Jr; Pannecouque, Christophe; De Clercq, Erik; Cushman, Mark

Investigation of the alkenyldiarylmethane non-nucleoside reverse transcriptase inhibitors as potential cAMP phosphodiesterase-4B2 inhibitors

研究烯基二芳基甲烷非核苷类逆转录酶抑制剂作为潜在的cAMP磷酸二酯酶-4B2抑制剂

Cullen, Matthew D; Cheung, York-Fong; Houslay, Miles D; Hartman, Tracy L; Watson, Karen M; Buckheit, Robert W Jr; Pannecouque, Christophe; De Clercq, Erik; Cushman, Mark