Re-engineering aryl methylcarbamates to confer high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase.
对芳基甲基氨基甲酸酯进行重新设计,使其对冈比亚按蚊抑制作用具有高选择性,而对人类乙酰胆碱酯酶则无此作用
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2012.05.103
Hartsel Joshua A, Wong Dawn M, Mutunga James M, Ma Ming, Anderson Troy D, Wysinski Ania, Islam Rafique, Wong Eric A, Paulson Sally L, Li Jianyong, Lam Polo C H, Totrov Maxim M, Bloomquist Jeffrey R, Carlier Paul R