Catalytic Degraders Effectively Address Kinase Site Mutations in EML4-ALK Oncogenic Fusions
催化降解剂可有效解决EML4-ALK致癌融合蛋白中的激酶位点突变
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c01864
Gao, Yang; Jiang, Baishan; Kim, Hellen; Berberich, Matthew J; Che, Jianwei; Donovan, Katherine A; Hatcher, John M; Huerta, Fidel; Kwiatkowski, Nicholas P; Liu, Yingpeng; Liuni, Peter P; Metivier, Rebecca J; Murali, Vineeth K; Nowak, Radosław P; Zhang, Tinghu; Fischer, Eric S; Gray, Nathanael S; Jones, Lyn H