日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Discovery of fully synthetic FKBP12-mTOR molecular glues

更正:发现了完全合成的FKBP12-mTOR分子胶

Deutscher, Robin C E; Meyners, Christian; Repity, Maximilian L; Sugiarto, Wisely Oki; Kolos, Jürgen M; Maciel, Edvaldo V S; Heymann, Tim; Geiger, Thomas M; Knapp, Stefan; Lermyte, Frederik; Hausch, Felix

Analgesia through FKBP51 inhibition at disease onset confers lasting relief from sensory and emotional chronic pain symptoms.

在疾病发作时通过抑制 FKBP51 来达到镇痛效果,可以持久缓解感觉和情绪方面的慢性疼痛症状。

Hestehave Sara, Florea Roxana, Singleton Samuel, Fedorec Alex J H, Caxaria Sara, Morgan Oakley B, Kopp Katharina Tatjana, Brown Laurence A, Heymann Tim, Sikandar Shafaq, Hausch Felix, Peirson Stuart N, Géranton Sandrine M

Novel PROTAC to target FKBP12: the potential to enhance bone morphogenetic protein activity and apoptosis in multiple myeloma.

新型 PROTAC 靶向 FKBP12:增强骨形态发生蛋白活性和多发性骨髓瘤细胞凋亡的潜力。

Quist-Lokken Ingrid, Tilseth Mira, Andersson-Rusch Clara, Hanif Md Abu, Walz Michael, Moen Johanna Fredrikke Nordstrand, Vik Megan Anne, Slordahl Tobias Schmidt, Sundan Anders, Hausch Felix, Holien Toril

Discovery of fully synthetic FKBP12-mTOR molecular glues

发现全合成的FKBP12-mTOR分子胶

Deutscher, Robin C E; Meyners, Christian; Repity, Maximilian L; Sugiarto, Wisely Oki; Kolos, Jürgen M; Maciel, Edvaldo V S; Heymann, Tim; Geiger, Thomas M; Knapp, Stefan; Lermyte, Frederik; Hausch, Felix

Exploring the potential of selective FKBP51 inhibitors on melanoma: an investigation of their in vitro and in vivo effects.

探索选择性 FKBP51 抑制剂对黑色素瘤的潜力:对其体外和体内效应的研究

Marrone Laura, Di Giacomo Valeria, Malasomma Chiara, Vecchione Marialuisa Alessandra, Hausch Felix, Cacace Massimiliano, D'Esposito Lucia, Tufano Martina, D'Arrigo Paolo, Romano Maria Fiammetta, Romano Simona

Targeting bacterial kinases as a strategy to counteract antibiotic resistance

以细菌激酶为靶点对抗抗生素耐药性

Buffa, Vanessa; Kowalewski, Julien; Qi, Guoman; Deutscher, Robin; Cica, Matijas; Richardoz, Marion; Tomaszczyk, Mathilde; Krämer, Andreas; Knapp, Stefan; Dunyach-Remy, Catherine; Rox, Katharina; Guichou, Jean-Francois; Lionne, Corinne; Hausch, Felix

Fragment-based drug design of a bacterial kinase inhibitor capable of increasing the antibiotic sensitivity of clinical isolates

基于片段的细菌激酶抑制剂药物设计,可提高临床分离株对抗生素的敏感性

Kowalewski, Julien; Deutscher, Robin; Richardoz, Marion; Tomaszczyk, Mathilde; Gelin, Muriel; Labesse, Gilles; Hausch, Felix; Wright, Gerard D; Dunyach-Remy, Catherine; Guichou, Jean-François; Lionne, Corinne

Cell-free tumor DNA analysis in advanced or metastatic breast cancer patients: mutation frequencies, testing intention, and clinical impact

晚期或转移性乳腺癌患者的无细胞肿瘤DNA分析:突变频率、检测目的和临床影响

Huebner, Hanna; Wimberger, Pauline; Laakmann, Elena; Ruckhäberle, Eugen; Ruebner, Matthias; Lehle, Sarah; Uhrig, Sabrina; Ziegler, Philipp; Link, Theresa; Hack, Carolin C; Belleville, Erik; Faull, Iris; Hausch, Marcus; Wallwiener, Diethelm; Schneeweiss, Andreas; Tesch, Hans; Brucker, Sara Y; Beckmann, Matthias W; Fasching, Peter A; Müller, Volkmar; Fehm, Tanja N

Phage therapy: Innovative approaches for refractory pulmonary infections

噬菌体疗法:治疗难治性肺部感染的创新方法

Dreizler, Johannes K; Meyners, Christian; Hausch, Felix; Qian, Yan; Zhu, Zhichen; Zhu, Jie; Chen, Liang; Du, Hong

Nondegradative Synthetic Molecular Glues Enter the Clinic

非降解性合成分子胶进入临床应用

Repity, Maximilian L; Deutscher, Robin C E; Hausch, Felix