日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Harmine Derivatives as Anticancer Agents Endowed With Potent and Selective Antileukemia Activity: Synthesis, Biological Evaluation, Proapoptotic and Genotoxic Activity

哈尔明衍生物作为具有强效选择性抗白血病活性的抗癌剂:合成、生物学评价、促凋亡和遗传毒性活性

Timbilla, Abdul Aziz; Pidany, Filip; Kohelova, Eliska; Kroustkova, Jana; Kralovec, Karel; Rataj, Jan; Ceckova, Martina; Maafi, Negar; Lopez, Víctor; Langa, Cristina Moliner; Kosturko, Stefan; Jenco, Jaroslav; Muthna, Darina; Koutova, Darja; Rezacova, Martina; Cahlikova, Lucie; Chlebek, Jakub; Havelek, Radim

Stemness and EMT profiles shift in xenografts derived from cisplatin-sensitive and cisplatin-tolerant ovarian cancer cells.

源自顺铂敏感和顺铂耐受卵巢癌细胞的异种移植瘤的干性和 EMT 特征发生了变化。

Mrkvicova Alena, Slavickova Marcela, Peterova Eva, Melounkova Lucie, Parova Helena, Havelek Radim, Krejcova Anna, Kohlerova Renata, Nekvindova Jana, Kazimirova Petra, Hajzlerova Milena, Rozkoš Tomáš, Rezacova Martina

Design of semisynthetic derivatives of the Amaryllidaceae alkaloid ambelline and exploration of their in vitro cytotoxic activities

设计石蒜科生物碱安贝林的半合成衍生物并探索其体外细胞毒活性

Ritomská, Aneta; Koutova, Darja; Křoustková, Jana; Královec, Karel; Muthná, Darina; Kuneš, Jiří; Nováková, Lucie; Havelek, Radim; Cahlíková, Lucie

Multimodal Contrast Agent Enabling pH Sensing Based on Organically Functionalized Gold Nanoshells with Mn-Zn Ferrite Cores

基于有机功能化金纳米壳和锰锌铁氧体核的多模态对比剂实现pH传感

Bui, Duong Thuy; Havelek, Radim; Královec, Karel; Kubíčková, Lenka; Kuličková, Jarmila; Matouš, Petr; Herynek, Vít; Kupčík, Jaroslav; Muthná, Darina; Řezanka, Pavel; Kaman, Ondřej

The Effect of Chronic Exposure of Graphene Nanoplates on the Viability and Motility of A549 Cells

石墨烯纳米片长期暴露对A549细胞活力和迁移能力的影响

Šestáková, Blanka; Schröterová, Ladislava; Bezrouk, Aleš; Čížková, Dana; Elkalaf, Moustafa; Havelek, Radim; Rudolf, Emil; Králová, Věra

Monoclonal anti-endoglin antibody TRC105 (carotuximab) prevents hypercholesterolemia and hyperglycemia-induced endothelial dysfunction in human aortic endothelial cells

单克隆抗内皮蛋白抗体 TRC105(卡罗妥昔单抗)可预防人主动脉内皮细胞高胆固醇血症和高血糖引起的内皮功能障碍

Katarina Tripska, Ivone Cristina Igreja Sá, Martina Vasinova, Matej Vicen, Radim Havelek, Samira Eissazadeh, Zuzana Svobodova, Barbora Vitverova, Charles Theuer, Carmelo Bernabeu, Petr Nachtigal

Disruption of Cell Adhesion and Cytoskeletal Networks by Thiol-Functionalized Silica-Coated Iron Oxide Nanoparticles

硫醇功能化二氧化硅包覆氧化铁纳米粒子对细胞粘附和细胞骨架网络的破坏作用

Královec, Karel; Melounková, Lucie; Slováková, Marcela; Mannová, Nikola; Sedlák, Miloš; Bartáček, Jan; Havelek, Radim

Substituted Piperazines as Novel Potential Radioprotective Agents

取代哌嗪类化合物作为新型潜在放射防护剂

Filipova, Alzbeta; Marek, Jan; Havelek, Radim; Pejchal, Jaroslav; Jelicova, Marcela; Cizkova, Jana; Majorosova, Martina; Muckova, Lubica; Kucera, Tomas; Prchal, Lukas; Psotka, Miroslav; Zivna, Natalie; Koutova, Darja; Sinkorova, Zuzana; Rezacova, Martina; Tichy, Ales

Chemical and Biological Aspects of Montanine-Type Alkaloids Isolated from Plants of the Amaryllidaceae Family

从石蒜科植物中分离得到的蒙塔宁型生物碱的化学和生物学特性

Koutová, Darja; Maafi, Negar; Havelek, Radim; Opletal, Lubomír; Blunden, Gerald; Řezáčová, Martina; Cahlíková, Lucie

Regulation and role of endoglin in cholesterol-induced endothelial and vascular dysfunction in vivo and in vitro

内皮因子在体内和体外胆固醇诱导的内皮和血管功能障碍中的调节和作用

Matej Vicen, Barbora Vitverova, Radim Havelek, Katerina Blazickova, Miloslav Machacek, Jana Rathouska, Iveta Najmanová, Eva Dolezelova, Alena Prasnicka, Magdalena Sternak, Carmelo Bernabeu, Petr Nachtigal