日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Correction to "From Discovery to Clinical Trial: YCT-529, an Oral NonHormonal Male Contraceptive Targeting the Retinoic Acid Receptor Alpha"

更正“从发现到临床试验：YCT-529，一种靶向视黄酸受体α的口服非激素男性避孕药”

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6c00520
Shi, Rui; Al Noman, Md Abdullah; Mannowetz, Nadja; Cheryala, Narsihmulu; Haque, Ehfazul; Taher, Noha; Maitra, Soma; Naqvi, Tahmina; Chung, Sanny S W; Bakshi, Akash; Hawkinson, Jon E; Wong, Henry L; Wolgemuth, Debra J; Georg, Gunda I
信号转导
免疫/内分泌
发表日期：2026
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From Discovery to Clinical Trial: YCT-529, an Oral NonHormonal Male Contraceptive Targeting the Retinoic Acid Receptor Alpha

从发现到临床试验：YCT-529，一种靶向视黄酸受体α的口服非激素男性避孕药

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c03051
Shi, Rui; Al Noman, Md Abdullah; Mannowetz, Nadja; Cheryala, Narsihmulu; Haque, Ehfazul; Maitra, Soma; Naqvi, Tahmina; Chung, Sanny S W; Bakshi, Akash; Hawkinson, Jon E; Wong, Henry L; Wolgemuth, Debra J; Georg, Gunda I
信号转导
免疫/内分泌
发表日期：2026
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Macrocyclic dihydropyridine analogs as pan-BET BD2-preferred inhibitors

大环二氢吡啶类似物作为泛BET BD2优先抑制剂

期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2025.117504
Jiang, Jiewei; Liang, Taimeng; Solberg, Jonathan; Chan, Alice; Kalra, Prakriti; Shi, Rui; Pomerantz, William C K; Hawkinson, Jon E; Schönbrunn, Ernst; Georg, Gunda I
发表日期：2025
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Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception

开发视黄酸受体α选择性拮抗剂作为新型男性避孕药的策略

期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2023.115821
Al Noman, Md Abdullah; Cuellar, Rebecca A D; Kyzer, Jillian L; Chung, Sanny S W; Cheryala, Narsihmulu; Holth, Trinh A D; Maitra, Soma; Naqvi, Tahmina; Wong, Henry L; Schönbrunn, Ernst; Hawkinson, Jon E; Wolgemuth, Debra J; Georg, Gunda I
信号转导
发表日期：2023
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Corrigendum: Discovery and Characterization of Multiple Classes of Human CatSper Blockers

更正：多种人类猫精子阻滞剂的发现和表征

期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.202200441
Carlson, Erick J; Francis, Rawle; Liu, Yutong; Li, Ping; Lyon, Maximilian; Santi, Celia M; Hook, Derek J; Hawkinson, Jon E; Georg, Gunda I
Human
发表日期：2022
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Steroidal Antagonists of Progesterone- and Prostaglandin E(1)-Induced Activation of the Cation Channel of Sperm

甾体拮抗剂可抑制孕酮和前列腺素E(1)诱导的精子阳离子通道激活

期刊:Molecular Pharmacology
影响因子:3
doi:10.1124/molpharm.121.000349
Carlson, Erick J; Georg, Gunda I; Hawkinson, Jon E
发表日期：2022
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Quantifying the Selectivity of Protein-Protein and Small Molecule Interactions with Fluorinated Tandem Bromodomain Reader Proteins

利用氟化串联溴结构域读取蛋白量化蛋白质-蛋白质和小分子相互作用的选择性

期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.0c00720
Kalra, Prakriti; McGraw, Logan; Kimbrough, Jennifer R; Pandey, Anil K; Solberg, Jonathan; Cui, Huarui; Divakaran, Anand; John, Kristen; Hawkinson, Jon E; Pomerantz, William C K
发表日期：2020
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Cooperativity Between Orthosteric Inhibitors and Allosteric Inhibitor 8-Anilino-1-Naphthalene Sulfonic Acid (ANS) in Cyclin-Dependent Kinase 2

细胞周期蛋白依赖性激酶2中正构抑制剂与变构抑制剂8-苯胺基-1-萘磺酸（ANS）的协同作用

期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.0c00169
Faber, Erik B; Tian, Defeng; Burban, David; Levinson, Nicholas M; Hawkinson, Jon E; Georg, Gunda I
信号转导
细胞生物学
发表日期：2020
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Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception

设计、合成并体外和体内评价乌本苷类似物作为强效选择性Na,K-ATPase α4亚型抑制剂用于男性避孕

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.7b00925
Syeda, Shameem Sultana; Sánchez, Gladis; Hong, Kwon Ho; Hawkinson, Jon E; Georg, Gunda I; Blanco, Gustavo
发表日期：2018
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Structure-Activity Studies of N-Butyl-1-deoxynojirimycin (NB-DNJ) Analogues: Discovery of Potent and Selective Aminocyclopentitol Inhibitors of GBA1 and GBA2

N-丁基-1-脱氧野尻霉素 (NB-DNJ) 类似物的构效关系研究：发现强效且选择性的 GBA1 和 GBA2 氨基环戊醇抑制剂

期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.201700558
Gu, Xingxian; Gupta, Vijayalaxmi; Yang, Yan; Zhu, Jin-Yi; Carlson, Erick J; Kingsley, Carolyn; Tash, Joseph S; Schönbrunn, Ernst; Hawkinson, Jon; Georg, Gunda I
发表日期：2017
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