日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MAVISp: A modular structure-based framework for protein variant effects

MAVISp:一种基于模块化结构的蛋白质变异效应框架

Arnaudi, Matteo; Utichi, Mattia; Degn, Kristine; Tiberti, Matteo; Beltrame, Ludovica; Krzesińska, Karolina; Besora, Pablo Sánchez-Izquierdo; Kiachaki, Eleni; Scrima, Simone; Bauer, Laura; Meldgård, Katrine; Melidi, Anna; Favaro, Lorenzo; Oswal, Anu; Tedeschi, Guglielmo; Dorčaková, Terézia; Estad, Alberte Heering; Breitenstein, Joachim; Safer, Jordan; Saridaki, Paraskevi; Sora, Valentina; Maselli, Francesca; Becker, Philipp; Vinhas, Jérémy; Pettenella, Alberto; Lambrughi, Matteo; Cava, Claudia; Rohlin, Anna; Nilbert, Mef; Iqbal, Sumaiya; Sackett, Peter Wad; Fas, Burcu Aykac; Papaleo, Elena

OGDHL promotes prostate cancer progression and regulates neuroendocrine marker expression and nucleotide abundance.

OGDHL促进前列腺癌进展,并调节神经内分泌标志物表达和核苷酸丰度。

Bernard Matthew J, Gallardo Andrea, Ruiz Angel, Diaz Johnny A, Nunley Nicholas M, Dove Rachel N, Zhang Shile, Lee Ernie, Heering Kylie Y, Varuzhanyan Grigor, Bopardikar Sachi, Hashimoto Takao, Agrawal Raag, Smith Chad M, Wilde Blake R, Matulionis Nedas, Richards Helen M, Lee Sandy Che-Eun S, Sharifi Marina N, Lang Joshua M, Zhao Shuang G, Witte Owen N, Haffner Michael C, Shackelford David B, Boutros Paul C, Christofk Heather R, Goldstein Andrew S

About a Trillion Times More Acidic than Expected? On the Difference Between the Hammett H(0) and the Unified pH Acidity of Sulfuric Acid

比预期酸度高出约一万亿倍?论硫酸的哈米特酸度 (H0) 与统一 pH 酸度之间的差异

Radtke, Valentin; Bäuerle, Monika; Stroh, Regina; Kienzle, Timo; Himmel, Daniel; Heering, Agnes; Nerut, Jaak; Lust, Enn; Leito, Ivo; Krossing, Ingo

Orphan G protein-coupled receptor GPRC5B controls macrophage function by facilitating prostaglandin E receptor 2 signaling

孤儿G蛋白偶联受体GPRC5B通过促进前列腺素E受体2信号传导来控制巨噬细胞功能

Jeonghyeon Kwon ,Haruya Kawase ,Kenny Mattonet ,Stefan Guenther ,Lisa Hahnefeld ,Jamal Shamsara ,Jan Heering ,Michael Kurz ,Sina Kirchhofer ,Cornelius Krasel ,Michaela Ulrich ,Margherita Persechino ,Sripriya Murthy ,Cesare Orlandi ,Christian D Sadik ,Gerd Geisslinger ,Moritz Bünemann ,Peter Kolb ,Stefan Offermanns ,Nina Wettschureck

The endocannabinoid anandamide mediates anti-inflammatory effects through activation of NR4A nuclear receptors.

内源性大麻素花生四烯酸乙醇胺通过激活 NR4A 核受体发挥抗炎作用

Teichmann Tom, Pflüger-Müller Beatrice, Giménez Virna Margarita Martín, Sailer Fiona, Dirks Henrik, Zehr Simonida, Warwick Timothy, Brettner Felix, Munoz-Tello Paola, Zimmer Andreas, Tegeder Irmgard, Thomas Dominique, Gurke Robert, Günther Stefan, Heering Jan, Proschak Ewgenij, Geisslinger Gerd, Bibli Iris-S, Heringdorf Dagmar Meyer Zu, Manucha Walter, Windbergs Maike, Knapp Stefan, Weigert Andreas, Leisegang Matthias S, Kojetin Douglas, Brandes Ralf P

Structure-Based Design of PROTACS for the Degradation of Soluble Epoxide Hydrolase.

基于结构的PROTACS设计用于降解可溶性环氧化物水解酶

Schönfeld Julia, Brunst Steffen, Ciomirtan Ludmila, Willmer Lena, Chromik Michel A, Kumar Adarsh, Froemel Timo, Liebisch Nick, Hackspacher Arne, Ehrler Johanna H M, Wintermeier Lukas, Hesse Christina, Fiedler Jan, Heering Jan, Freitag Hinrich, Zardo Patrick, Fieguth Hans-Gerd, Brüggerhoff Astrid, Jakob Josefine, Häupl Björn, Weizel Lilia, Kaiser Astrid, Schubert-Zsilavecz Manfred, Oellerich Thomas, Fleming Ingrid, Schebb Nils H, Fürst Robert, Kannt Aimo, Knapp Stefan, Proschak Ewgenij, Hiesinger Kerstin

Structural and mechanistic profiling of Nurr1 modulation by vidofludimus enables structure-guided ligand design

通过对维多氟替卡松调控Nurr1的结构和机制进行分析,可以实现结构导向的配体设计。

López-García, Úrsula; Vietor, Jan; Marschner, Julian A; Heering, Jan; Morozov, Vasily; Wein, Thomas; Merk, Daniel

Ethical considerations on the use of big data and artificial intelligence in kidney research from the ERA ethics committee

欧洲肾脏病研究协会(ERA)伦理委员会关于在肾脏研究中使用大数据和人工智能的伦理考量

Van Biesen, Wim; Ponikvar, Jadranka Buturovic; Fontana, Monica; Heering, Peter; Sever, Mehmet S; Sawhney, Simon; Luyckx, Valerie

S1PR4-dependent effects of Etrasimod on primary human myeloid immune cell activation

Etrasimod 对原代人髓系免疫细胞活化的 S1PR4 依赖性效应

Sailer, Fiona K; Palmer, Megan A; Aliraj, Blerina; Heering, Jan; Brockmann, Andreas; Elewa, Mohammed A F; Röhrig, Aissa; Proschak, Ewgenij; Stepniak, Dariusz T; Ramsey, Simeon; Brüne, Bernhard; Weigert, Andreas

Universal Reversible Hydrogen Potential for Electrocatalytic Ammonia Splitting Reactions in Nonaqueous Solvents from Unified pH Measurements

基于统一pH测量的非水溶剂中电催化氨分解反应的通用可逆氢电位

Mi, Chenjia; Saame, Jaan; Heering, Agnes; Zhang, Xiaoyin; Abubakar, Oluwafemi; Leito, Ivo; Hamann, Thomas W