日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Perspective change: Students as instructors - a report of experiences by nursing and medical students in the role of peer tutors

视角转变:学生担任教师——护理和医学生担任同伴辅导员的经验报告

Frei, Patrick; Fischer, Tim; Heering, Jan-Ole; Gutmann, Sarah

The endocannabinoid anandamide mediates anti-inflammatory effects through activation of NR4A nuclear receptors.

内源性大麻素花生四烯酸乙醇胺通过激活 NR4A 核受体发挥抗炎作用

Teichmann Tom, Pflüger-Müller Beatrice, Giménez Virna Margarita Martín, Sailer Fiona, Dirks Henrik, Zehr Simonida, Warwick Timothy, Brettner Felix, Munoz-Tello Paola, Zimmer Andreas, Tegeder Irmgard, Thomas Dominique, Gurke Robert, Günther Stefan, Heering Jan, Proschak Ewgenij, Geisslinger Gerd, Bibli Iris-S, Heringdorf Dagmar Meyer Zu, Manucha Walter, Windbergs Maike, Knapp Stefan, Weigert Andreas, Leisegang Matthias S, Kojetin Douglas, Brandes Ralf P

Structure-Based Design of PROTACS for the Degradation of Soluble Epoxide Hydrolase.

基于结构的PROTACS设计用于降解可溶性环氧化物水解酶

Schönfeld Julia, Brunst Steffen, Ciomirtan Ludmila, Willmer Lena, Chromik Michel A, Kumar Adarsh, Froemel Timo, Liebisch Nick, Hackspacher Arne, Ehrler Johanna H M, Wintermeier Lukas, Hesse Christina, Fiedler Jan, Heering Jan, Freitag Hinrich, Zardo Patrick, Fieguth Hans-Gerd, Brüggerhoff Astrid, Jakob Josefine, Häupl Björn, Weizel Lilia, Kaiser Astrid, Schubert-Zsilavecz Manfred, Oellerich Thomas, Fleming Ingrid, Schebb Nils H, Fürst Robert, Kannt Aimo, Knapp Stefan, Proschak Ewgenij, Hiesinger Kerstin

Structural and mechanistic profiling of Nurr1 modulation by vidofludimus enables structure-guided ligand design

通过对维多氟替卡松调控Nurr1的结构和机制进行分析,可以实现结构导向的配体设计。

López-García, Úrsula; Vietor, Jan; Marschner, Julian A; Heering, Jan; Morozov, Vasily; Wein, Thomas; Merk, Daniel

S1PR4-dependent effects of Etrasimod on primary human myeloid immune cell activation

Etrasimod 对原代人髓系免疫细胞活化的 S1PR4 依赖性效应

Sailer, Fiona K; Palmer, Megan A; Aliraj, Blerina; Heering, Jan; Brockmann, Andreas; Elewa, Mohammed A F; Röhrig, Aissa; Proschak, Ewgenij; Stepniak, Dariusz T; Ramsey, Simeon; Brüne, Bernhard; Weigert, Andreas

Fragment-Based Discovery of Drug-like LRH-1 Agonists

基于片段的类药LRH-1激动剂发现

Lang, Alisa; Ildefeld, Niklas; Lillich, Felix F; Kaiser, Astrid; Busch, Romy; Marschner, Julian A; Proschak, Ewgenij; Heering, Jan; Schubert-Zsilavecz, Manfred; Merk, Daniel

Fatty Acid Mimetic Fragments as Liver Receptor Homologue-1 Modulators

脂肪酸模拟片段作为肝脏受体同源物-1调节剂

Lang, Alisa; Stiller, Tanja; Ildefeld, Niklas; Heitel, Pascal; Isigkeit, Laura; Proschak, Ewgenij; Heering, Jan; Schubert-Zsilavecz, Manfred; Merk, Daniel

Optimization and Evaluation of Complementary Degrader Discovery Assays for Application in Screening.

优化和评价互补降解剂发现试验在筛选中的应用

Huchting Johanna, Weller Arjen, Schweizer Moyra, Brandt Mona, Heering Jan, Kuzikov Maria, Wolf Markus, Reinshagen Jeanette, Queisser Markus A, Gribbon Philip, Zaliani Andrea, Pless Ole, Kannt Aimo

Development of a Potent and Selective G2A (GPR132) Agonist.

开发一种高效选择性的G2A(GPR132)激动剂

Hernandez-Olmos Victor, Heering Jan, Marinescu Beatrice, Schermeng Tina, Ivanov Vladimir V, Moroz Yurii S, Nevermann Sheila, Mathes Marius, Ehrler Johanna H M, Alnouri Mohamad Wessam, Wolf Markus, Haydo Alicia S, Schmachtel Tessa, Zaliani Andrea, Höfner Georg, Kaiser Astrid, Schubert-Zsilavecz Manfred, Beck-Sickinger Annette G, Offermanns Stefan, Gribbon Philipp, Rieger Michael A, Merk Daniel, Sisignano Marco, Steinhilber Dieter, Proschak Ewgenij

Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPARγ Modulation

靶向替代维生素E代谢物结合位点可实现非经典PPARγ调节

Arifi, Silvia; Marschner, Julian A; Pollinger, Julius; Isigkeit, Laura; Heitel, Pascal; Kaiser, Astrid; Obeser, Lennart; Höfner, Georg; Proschak, Ewgenij; Knapp, Stefan; Chaikuad, Apirat; Heering, Jan; Merk, Daniel