An Optimized Dihydrodibenzothiazepine Lead Compound (SBI-0797750) as a Potent and Selective Inhibitor of Plasmodium falciparum and P. vivax Glucose 6-Phosphate Dehydrogenase 6-Phosphogluconolactonase
优化的二氢二苯并硫氮卓类先导化合物 (SBI-0797750) 可作为恶性疟原虫和间日疟原虫葡萄糖 6-磷酸脱氢酶 6-磷酸葡萄糖酸内酯酶的强效选择性抑制剂
期刊:Antimicrobial Agents and Chemotherapy
影响因子:4.1
doi:10.1128/aac.02109-21
Isabell Berneburg #, Satyamaheshwar Peddibhotla #, Kim C Heimsch, Kristina Haeussler, Patrick Maloney, Palak Gosalia, Janina Preuss, Mahsa Rahbari, Oleksii Skorokhod, Elena Valente, Daniela Ulliers, Luigi Felice Simula, Kathrin Buchholz, Michael P Hedrick, Paul Hershberger, Thomas D Y Chung, Michael