日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of spirodioxolane nsP2 helicase inhibitors with antialphaviral activity

鉴定具有抗甲病毒活性的螺二氧戊环nsP2解旋酶抑制剂

Oh, Hans J; Sears, John D; Ramalingam, Bose Muthu; Saleem, Rahman Shah Zaib; Davis-Gilbert, Zachary W; Hossain, Mohammed Anwar; Moorman, Stella R; Ohja, Durbadal; Martinez, Sabian A; Burdick, Jane E; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Todd, Matthew H; Willson, Timothy M

Broadly active intranasal influenza vaccine with a nanocomplex particulate adjuvant targeting mast cells and toll-like receptor 9

一种广谱活性鼻内流感疫苗,含有靶向肥大细胞和 Toll 样受体 9 的纳米复合物颗粒佐剂

Ontiveros-Padilla, Luis; Hendy, Dylan A; Pena, Erik S; Williamson, Grace L; Murphy, Connor T; Lukesh, Nicole R; Ashcraft, Kathleen A; Abraham, Mathew A; Landon, Chelsea D; Staats, Herman F; Abraham, Soman N; Carlock, Michael; Ross, Ted M; Petrovsky, Nikolai; Heise, Mark T; Bachelder, Eric M; Ainslie, Kristy M

Identification of Direct-Acting nsP2 Helicase Inhibitors with Antialphaviral Activity

鉴定具有抗甲病毒活性的直接作用nsP2解旋酶抑制剂

Muthu Ramalingam, Bose; Sears, John D; Talbot, Kacey M; Su, Yuan-Wei Norman; Houliston, Scott; Hossain, Mohammed Anwar; Davis-Gilbert, Zachary W; Zhao, Chunqing; Oh, Hans J; Brown, Peter J; Sanders, Marcia K; Moorman, Stella R; Ojha, Durbadal; Burdick, Jane E; Law, Isabella; Morales, Noah L; Martinez, Sabian A; Loppnau, Peter; Garcia Perez, Julia; Drobish, Adam M; Morrison, Thomas E; Streblow, Zachary J; Streblow, Daniel N; Arrowsmith, Cheryl H; Vargason, Ava; Couñago, Rafael M; Halabelian, Levon; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

N-Alkyl Sulfamates as a New Class of nsP2 Cysteine Protease Inhibitors with Broad-Spectrum Antialphaviral Activity

N-烷基氨基磺酸酯作为一类新型nsP2半胱氨酸蛋白酶抑制剂,具有广谱抗甲病毒活性

Ghoshal, Anirban; Sears, John D; Hossain, Mohammad Anwar; Tse, Edwin G; Howell, Stefanie; Burdick, Jane E; Morales, Noah L; Martinez, Sabian A; Law, Isabella; Streblow, Zachary J; Streblow, Daniel N; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Species-Dependent Metabolism of a Covalent nsP2 Protease Inhibitor with In Vivo Antialphaviral Activity.

具有体内抗甲病毒活性的共价nsP2蛋白酶抑制剂的物种依赖性代谢

Hossain Mohammad Anwar, Mayo Abigail K, Ghoshal Anirban, Taft-Benz Sharon, Anderson Elizabeth, Morales Noah L, Pressey Katia D, Vargason Ava, Brouwer Kim L R, Moorman Nathaniel J, Heise Mark T, Willson Timothy M

Enantioselective Chemical Probe for Chikungunya nsP2 Helicase with Antialphaviral Activity

具有抗甲病毒活性的基孔肯雅病毒nsP2解旋酶对映选择性化学探针

Muthu Ramalingam, Bose; Oh, Hans J; Sears, John D; Chen, Chun-Hsing; Vala, Anand; Liu, Shubin; Talbot, Kacey M; Hossain, Mohammed Anwar; Brown, Peter J; Houliston, Scott; Garcia Perez, Julia; Li, Fengling; Amare, Meareg G; Halfmann, Peter; Smith, Jessica L; Hirsch, Alec J; Arrowsmith, Cheryl H; Halabelian, Levon; Vargason, Ava; Couñago, Rafael M; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Development of a virulent O'nyong'nyong challenge model to determine heterologous protection mediated by a hydrogen peroxide-inactivated chikungunya virus vaccine

建立强毒性O'nyong'nyong病毒攻击模型,以确定过氧化氢灭活的基孔肯雅病毒疫苗介导的异源保护作用

Weber, Whitney C; Streblow, Zachary J; Andoh, Takeshi F; Denton, Michael; Raué, Hans-Peter; Amanna, Ian J; Slifka, Dawn K; Kreklywich, Craig N; Arduino, Irene; Sulgey, Gauthami; Streblow, Magdalene M; Heise, Mark T; Slifka, Mark K; Streblow, Daniel N

Insulin deficiency inhibits vaccine-mediated antibody and germinal center B-cell formation in mice

胰岛素缺乏会抑制小鼠疫苗介导的抗体和生发中心B细胞的形成。

Genito, Christopher J; Ariel, Pablo; Heise, Mark T; Thurlow, Lance R

Novel Computational Pipeline to Identify Target Sites for Broad Spectrum Antiviral Drugs

用于识别广谱抗病毒药物靶点的新型计算流程

Sears, John D; Popov, Konstantin I; Sylvester, Paul; Dickmander, Rebekah; Loome-Diaz, Jennifer; Chang, Che-Kang; Huff, Julia; Sanders, Wes; Saba, Nicholas A; Sorensen, Madeleine; Drobish, Adam M; May, Nicholas A; Namitz, Kevin; Fecko, Julia; Arnold, Jamie J; Yennawar, Neela H; Cameron, Craig E; Morrison, Thomas E; Tropsha, Alexander; Heise, Mark T; Moorman, Nathaniel J

Myeloperoxidase-ANCA IgG induces different forms of small vessel vasculitis based on type of synergistic immune stimuli.

髓过氧化物酶-ANCA IgG 根据协同免疫刺激的类型诱发不同形式的小血管炎

Hu Peiqi, Xiao Hong, Alba Marco A, Atkins Hannah M, Gou Shenju, Hu Yanglin, Gomez John C, Jania Corey M, Martin Jessica R, Morrison Thomas E, Tilley Stephen L, Heise Mark T, Doerschuk Claire M, Falk Ronald J, Jennette J Charles