日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulphostin-inspired N-phosphonopiperidones as selective covalent DPP8 and DPP9 inhibitors.

受磺基膦酸酯启发而合成的 N-膦酸哌啶酮类化合物作为选择性共价 DPP8 和 DPP9 抑制剂

Sewald Leonard, Tabak Werner W A, Fehr Lorenz, Zolg Samuel, Najdzion Maja, Verhoef Carlo J A, Podlesainski David, Geiss-Friedlander Ruth, Lammens Alfred, Kaschani Farnusch, Hellerschmied Doris, Huber Robert, Kaiser Markus

Conformational plasticity of a BiP-GRP94 chaperone complex

BiP-GRP94分子伴侣复合物的构象可塑性

Brenner, Joel Cyrille; Zirden, Linda Charlotte; Buzuk, Lana; Almeida-Hernandez, Yasser; Radzuweit, Lea; Diamantino, Joao; Kaschani, Farnusch; Kaiser, Markus; Sanchez-Garcia, Elsa; Poepsel, Simon; Hellerschmied, Doris

The serine protease HTRA1 targets tau fibrils and provides a proteolytic barrier against pathogenic protein conformations

丝氨酸蛋白酶HTRA1靶向tau蛋白原纤维,并提供一道蛋白水解屏障,抵御致病性蛋白构象的形成。

Hagemeier, Birte; Ripkens, Kamilla; Schulze, Nina; Bluemke, Anika; Strzala, Michal; Koci, Michelle; Kaschani, Farnusch; Kaiser, Markus; Erkelenz, Michael; Schluecker, Sebastian; Merdanovic, Melisa; Poepsel, Simon; Hellerschmied, Doris; Burston, Steven G; Ehrmann, Michael

A Photocaged N-Phosphonopiperidinone as a Selective Photo-Cleavable DPP8/9 Inhibitor

一种光笼状N-膦哌啶酮作为选择性光裂解DPP8/9抑制剂

Sewald, Leonard; Molke, Niko; Tabak, Werner W A; Haak, Anette; Najdzion, Maja; Geiss-Friedlander, Ruth; Hellerschmied, Doris; Huber, Robert; Kaiser, Markus

Ubiquitin-mediated degradation at the Golgi apparatus

高尔基体中的泛素介导降解

Buzuk, Lana; Hellerschmied, Doris

Modular PROTAC Design for the Degradation of Oncogenic BCR-ABL

用于降解致癌性 BCR-ABL 的模块化 PROTAC 设计

Lai, Ashton C; Toure, Momar; Hellerschmied, Doris; Salami, Jemilat; Jaime-Figueroa, Saul; Ko, Eunhwa; Hines, John; Crews, Craig M

The Nuclear Pore-Associated TREX-2 Complex Employs Mediator to Regulate Gene Expression

核孔相关TREX-2复合物利用介导因子调控基因表达

Schneider, Maren; Hellerschmied, Doris; Schubert, Tobias; Amlacher, Stefan; Vinayachandran, Vinesh; Reja, Rohit; Pugh, B Franklin; Clausen, Tim; Köhler, Alwin