日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis, Biological Evaluation, and Docking Studies of Antagonistic Hydroxylated Arecaidine Esters Targeting mAChRs

针对 mAChRs 的拮抗性羟基化槟榔碱酯的合成、生物学评价及对接研究

Jonas Kilian, Marlon Millard, Marius Ozenil, Dominik Krause, Khadija Ghaderi, Wolfgang Holzer, Ernst Urban, Helmut Spreitzer, Wolfgang Wadsak, Marcus Hacker, Thierry Langer, Verena Pichler

Discovery of melanin-concentrating hormone receptor 1 in brown adipose tissue

棕色脂肪组织中发现黑色素浓缩激素受体 1

Cécile Philippe, Eva-Maria Klebermass, Theresa Balber, Oana C Kulterer, Markus Zeilinger, Gerda Egger, Monika Dumanic, Carsten T Herz, Florian W Kiefer, Christian Scheuba, Thomas Scherer, Clemens Fürnsinn, Chrysoula Vraka, Katharina Pallitsch, Helmut Spreitzer, Wolfgang Wadsak, Helmut Viernstein, Ma

Synthesis, Biological, and Computational Evaluation of Antagonistic, Chiral Hydrobenzoin Esters of Arecaidine Targeting mAChR M1

针对 mAChR M1 的拮抗性手性槟榔氢苯甲酸酯的合成、生物学和计算评估

Marius Ozenil, Jonas Aronow, Daniela Piljak, Chrysoula Vraka, Wolfgang Holzer, Helmut Spreitzer, Wolfgang Wadsak, Marcus Hacker, Verena Pichler

SNAPshots of the MCHR1: a Comparison Between the PET-Tracers [18F]FE@SNAP and [11C]SNAP-7941

MCHR1 的快照:PET 示踪剂 [18F]FE@SNAP 与 [11C]SNAP-7941 之间的比较

Cécile Philippe, Markus Zeilinger, Monika Dumanic, Florian Pichler, Lukas Fetty, Chrysoula Vraka, Theresa Balber, Wolfgang Wadsak, Katharina Pallitsch, Helmut Spreitzer, Rupert Lanzenberger, Marcus Hacker, Markus Mitterhauser

In vitro Radiopharmaceutical Evidence for MCHR1 Binding Sites in Murine Brown Adipocytes

小鼠棕色脂肪细胞中 MCHR1 结合位点的体外放射性药物证据

Theresa Balber, Katarína Benčurová, Florian Wolfgang Kiefer, Oana Cristina Kulterer, Eva-Maria Klebermass, Gerda Egger, Loan Tran, Karl-Heinz Wagner, Helmut Viernstein, Katharina Pallitsch, Helmut Spreitzer, Marcus Hacker, Wolfgang Wadsak, Markus Mitterhauser, Cécile Philippe

In vivo evaluation of radiotracers targeting the melanin-concentrating hormone receptor 1: [11C]SNAP-7941 and [18F]FE@SNAP reveal specific uptake in the ventricular system

针对黑色素浓缩激素受体 1 的放射性示踪剂的体内评估:[11C]SNAP-7941 和 [18F]FE@SNAP 揭示了心室系统中的特定摄取

Markus Zeilinger, Monika Dumanic, Florian Pichler, Lubos Budinsky, Wolfgang Wadsak, Katharina Pallitsch, Helmut Spreitzer, Rupert Lanzenberger, Marcus Hacker, Markus Mitterhauser, Cécile Philippe2

New approaches for the reliable in vitro assessment of binding affinity based on high-resolution real-time data acquisition of radioligand-receptor binding kinetics

基于放射性配体-受体结合动力学的高分辨率实时数据采集的可靠体外评估结合亲和力的新方法

Markus Zeilinger, Florian Pichler, Lukas Nics, Wolfgang Wadsak, Helmut Spreitzer, Marcus Hacker, Markus Mitterhauser