日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of potent small-molecule inhibitors of lipoprotein(a) formation

发现有效的脂蛋白(a)形成小分子抑制剂

Nuria Diaz, Carlos Perez, Ana Maria Escribano, Gema Sanz, Julian Priego, Celia Lafuente, Mario Barberis, Luis Calle, Juan Felix Espinosa, Birgit T Priest, Hong Y Zhang, Amanda K Nosie, Joseph V Haas, Ellen Cannady, Anthony Borel, Albert E Schultze, J Michael Sauder, Jörg Hendle, Ken Weichert, Stephe

Discovery and clinical translation of ceperognastat, an O-GlcNAcase (OGA) inhibitor, for the treatment of Alzheimer's disease

发现并临床转化了 O-GlcNAcase (OGA) 抑制剂 ceperognastat 用于治疗阿尔茨海默病

Kielbasa, William; Goldsmith, Paul; Donnelly, Kevin B; Nuthall, Hugh N; Shcherbinin, Sergey; Fleisher, Adam S; Hendle, Jörg; DuBois, Susan L; Lowe, Stephen L; Zhang, Feiyu Fred; Woerly, Eric M; Dreyfus, Nicolas J-F; Evans, David; Gilmore, Jeremy; Mancini, Michele; Constantinescu, Cristian C; Gunn, Roger N; Russell, David S; Collins, Emily C; Brys, Miroslaw; Hutton, Michael L; Mergott, Dustin J

Epitope topography of agonist antibodies to the checkpoint inhibitory receptor BTLA

检查点抑制受体BTLA激动剂抗体的表位拓扑结构

Cheung, Timothy C; Atwell, Shane; Bafetti, Lisa; Cuenca, Paulina Delgado; Froning, Karen; Hendle, Jorg; Hickey, Michael; Ho, Carolyn; Huang, Jiawen; Lieu, Ricky; Lim, Stacie; Lippner, David; Obungu, Victor; Ward-Kavanagh, Lindsay; Weichert, Kenneth; Ware, Carl F; Vendel, Andrew C

Idea2Data: Toward a New Paradigm for Drug Discovery

Idea2Data:迈向药物发现的新范式

Nicolaou, Christos A; Humblet, Christine; Hu, Hong; Martin, Eva M; Dorsey, Frank C; Castle, Thomas M; Burton, Keith Ian; Hu, Haitao; Hendle, Jorg; Hickey, Michael J; Duerksen, Joel; Wang, Jibo; Erickson, Jon A

Computational design of a specific heavy chain/κ light chain interface for expressing fully IgG bispecific antibodies

用于表达完全 IgG 双特异性抗体的特定重链/κ 轻链界面的计算设计

K J Froning, A Leaver-Fay, X Wu, S Phan, L Gao, F Huang, A Pustilnik, M Bacica, K Houlihan, Q Chai, J R Fitchett, J Hendle, B Kuhlman, S J Demarest

Outcome of the First wwPDB/CCDC/D3R Ligand Validation Workshop

第一次 wwPDB/CCDC/D3R 配体验证研讨会成果

Adams, Paul D; Aertgeerts, Kathleen; Bauer, Cary; Bell, Jeffrey A; Berman, Helen M; Bhat, Talapady N; Blaney, Jeff M; Bolton, Evan; Bricogne, Gerard; Brown, David; Burley, Stephen K; Case, David A; Clark, Kirk L; Darden, Tom; Emsley, Paul; Feher, Victoria A; Feng, Zukang; Groom, Colin R; Harris, Seth F; Hendle, Jorg; Holder, Thomas; Joachimiak, Andrzej; Kleywegt, Gerard J; Krojer, Tobias; Marcotrigiano, Joseph; Mark, Alan E; Markley, John L; Miller, Matthew; Minor, Wladek; Montelione, Gaetano T; Murshudov, Garib; Nakagawa, Atsushi; Nakamura, Haruki; Nicholls, Anthony; Nicklaus, Marc; Nolte, Robert T; Padyana, Anil K; Peishoff, Catherine E; Pieniazek, Susan; Read, Randy J; Shao, Chenghua; Sheriff, Steven; Smart, Oliver; Soisson, Stephen; Spurlino, John; Stouch, Terry; Svobodova, Radka; Tempel, Wolfram; Terwilliger, Thomas C; Tronrud, Dale; Velankar, Sameer; Ward, Suzanna C; Warren, Gregory L; Westbrook, John D; Williams, Pamela; Yang, Huanwang; Young, Jasmine

SGX523 is an exquisitely selective, ATP-competitive inhibitor of the MET receptor tyrosine kinase with antitumor activity in vivo

SGX523 是一种选择性极好的 ATP 竞争性 MET 受体酪氨酸激酶抑制剂,具有体内抗肿瘤活性

Sean G Buchanan, Jorg Hendle, Patrick S Lee, Christopher R Smith, Pierre-Yves Bounaud, Katti A Jessen, Crystal M Tang, Nanni H Huser, Jeremy D Felce, Karen J Froning, Marshall C Peterman, Brandon E Aubol, Steve F Gessert, J Michael Sauder, Kenneth D Schwinn, Marijane Russell, Isabelle A Rooney, Jaso

Deposit3D: a tool for automating structure depositions to the Protein Data Bank

Deposit3D:一种用于自动向蛋白质数据库提交结构信息的工具

Badger, J; Hendle, J; Burley, S K; Kissinger, C R

A review of immunofluorescent patterns associated with antineutrophil cytoplasmic antibodies (ANCA) and their differentiation from other antibodies

对与抗中性粒细胞胞浆抗体 (ANCA) 相关的免疫荧光模式及其与其他抗体的鉴别诊断进行综述

Savige, J A; Paspaliaris, B; Silvestrini, R; Davies, D; Nikoloutsopoulos, T; Sturgess, A; Neil, J; Pollock, W; Dunster, K; Hendle, M