日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Differential roles of putative arginine fingers of AAA(+) ATPases Rvb1 and Rvb2.

AAA(+) ATPases Rvb1 和 Rvb2 的假定精氨酸指的不同作用

Warnock Jennifer L, Ball Jacob A, Najmi Saman M, Henes Mina, Vazquez Amanda, Koshnevis Sohail, Wieden Hans-Joachim, Conn Graeme L, Ghalei Homa

Deciphering the Molecular Mechanism of HCV Protease Inhibitor Fluorination as a General Approach to Avoid Drug Resistance

解析HCV蛋白酶抑制剂氟化作用的分子机制,是避免耐药性的通用方法

Zephyr, Jacqueto; Nageswara Rao, Desaboini; Vo, Sang V; Henes, Mina; Kosovrasti, Klajdi; Matthew, Ashley N; Hedger, Adam K; Timm, Jennifer; Chan, Elise T; Ali, Akbar; Kurt Yilmaz, Nese; Schiffer, Celia A

Drug Design Strategies to Avoid Resistance in Direct-Acting Antivirals and Beyond

避免直接抗病毒药物及其他药物产生耐药性的药物设计策略

Matthew, Ashley N; Leidner, Florian; Lockbaum, Gordon J; Henes, Mina; Zephyr, Jacqueto; Hou, Shurong; Rao, Desaboini Nageswara; Timm, Jennifer; Rusere, Linah N; Ragland, Debra A; Paulsen, Janet L; Prachanronarong, Kristina; Soumana, Djade I; Nalivaika, Ellen A; Kurt Yilmaz, Nese; Ali, Akbar; Schiffer, Celia A

Discovery of Quinoxaline-Based P1-P3 Macrocyclic NS3/4A Protease Inhibitors with Potent Activity against Drug-Resistant Hepatitis C Virus Variants

发现对耐药性丙型肝炎病毒变异株具有强效活性的喹喔啉类P1-P3大环NS3/4A蛋白酶抑制剂

Nageswara Rao, Desaboini; Zephyr, Jacqueto; Henes, Mina; Chan, Elise T; Matthew, Ashley N; Hedger, Adam K; Conway, Hasahn L; Saeed, Mohsan; Newton, Alicia; Petropoulos, Christos J; Huang, Wei; Kurt Yilmaz, Nese; Schiffer, Celia A; Ali, Akbar

Pan-3C Protease Inhibitor Rupintrivir Binds SARS-CoV-2 Main Protease in a Unique Binding Mode

泛3C蛋白酶抑制剂鲁平替韦以独特的结合模式与SARS-CoV-2主蛋白酶结合

Lockbaum, Gordon J; Henes, Mina; Lee, Jeong Min; Timm, Jennifer; Nalivaika, Ellen A; Thompson, Paul R; Kurt Yilmaz, Nese; Schiffer, Celia A

Molecular and Structural Mechanism of Pan-Genotypic HCV NS3/4A Protease Inhibition by Glecaprevir

格卡瑞韦抑制泛基因型HCV NS3/4A蛋白酶的分子和结构机制

Timm, Jennifer; Kosovrasti, Klajdi; Henes, Mina; Leidner, Florian; Hou, Shurong; Ali, Akbar; Kurt Yilmaz, Nese; Schiffer, Celia A