日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Whole Ovary Immunofluorescence, Clearing, and Multiphoton Microscopy for Quantitative 3D Analysis of the Developing Ovarian Reserve in Mouse.

小鼠卵巢发育储备的定量三维分析:全卵巢免疫荧光、透明化和多光子显微镜技术

Boateng Ruby, Boechat Nathaniel, Henrich Philipp P, Bolcun-Filas Ewelina

Global Spread of Mutant PfCRT and Its Pleiotropic Impact on Plasmodium falciparum Multidrug Resistance and Fitness

突变型PfCRT的全球传播及其对恶性疟原虫多药耐药性和适应性的多效性影响

Dhingra, Satish K; Gabryszewski, Stanislaw J; Small-Saunders, Jennifer L; Yeo, Tomas; Henrich, Philipp P; Mok, Sachel; Fidock, David A

A Variant PfCRT Isoform Can Contribute to Plasmodium falciparum Resistance to the First-Line Partner Drug Piperaquine

PfCRT 同工酶的变异可能导致恶性疟原虫对一线联合药物哌喹产生耐药性

Dhingra, Satish K; Redhi, Devasha; Combrinck, Jill M; Yeo, Tomas; Okombo, John; Henrich, Philipp P; Cowell, Annie N; Gupta, Purva; Stegman, Matthew L; Hoke, Jonathan M; Cooper, Roland A; Winzeler, Elizabeth; Mok, Sachel; Egan, Timothy J; Fidock, David A

Evolution of Fitness Cost-Neutral Mutant PfCRT Conferring P. falciparum 4-Aminoquinoline Drug Resistance Is Accompanied by Altered Parasite Metabolism and Digestive Vacuole Physiology

赋予恶性疟原虫4-氨基喹啉类药物耐药性的适应性成本中性突变体PfCRT的进化伴随着寄生虫代谢和消化液泡生理的改变

Gabryszewski, Stanislaw J; Dhingra, Satish K; Combrinck, Jill M; Lewis, Ian A; Callaghan, Paul S; Hassett, Matthew R; Siriwardana, Amila; Henrich, Philipp P; Lee, Andrew H; Gnädig, Nina F; Musset, Lise; Llinás, Manuel; Egan, Timothy J; Roepe, Paul D; Fidock, David A

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

三氨基嘧啶是一种速效且长效的抗疟疾候选药物。

Hameed P, Shahul; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P; Magistrado, Pamela A; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Roy Choudhury, Nilanjana; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K R; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Jiménez-Díaz, María Belén; Martínez, María Santos; Sanz, Laura María; Coburn-Flynn, Olivia; Fidock, David A; Lukens, Amanda K; Wirth, Dyann F; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K

Balancing drug resistance and growth rates via compensatory mutations in the Plasmodium falciparum chloroquine resistance transporter

通过恶性疟原虫氯喹耐药转运蛋白的补偿性突变来平衡耐药性和生长速率

Petersen, Ines; Gabryszewski, Stanislaw J; Johnston, Geoffrey L; Dhingra, Satish K; Ecker, Andrea; Lewis, Rebecca E; de Almeida, Mariana Justino; Straimer, Judith; Henrich, Philipp P; Palatulan, Eugene; Johnson, David J; Coburn-Flynn, Olivia; Sanchez, Cecilia; Lehane, Adele M; Lanzer, Michael; Fidock, David A

Evidence for pyronaridine as a highly effective partner drug for treatment of artemisinin-resistant malaria in a rodent model

在啮齿动物模型中,吡咯萘啶作为治疗青蒿素耐药疟疾的高效辅助药物的证据

Henrich, Philipp P; O'Brien, Connor; Sáenz, Fabián E; Cremers, Serge; Kyle, Dennis E; Fidock, David A

Quinine dimers are potent inhibitors of the Plasmodium falciparum chloroquine resistance transporter and are active against quinoline-resistant P. falciparum

奎宁二聚体是恶性疟原虫氯喹耐药转运蛋白的强效抑制剂,对喹啉耐药的恶性疟原虫有效。

Hrycyna, Christine A; Summers, Robert L; Lehane, Adele M; Pires, Marcos M; Namanja, Hilda; Bohn, Kelsey; Kuriakose, Jerrin; Ferdig, Michael; Henrich, Philipp P; Fidock, David A; Kirk, Kiaran; Chmielewski, Jean; Martin, Rowena E

A key role for lipoic acid synthesis during Plasmodium liver stage development.

硫辛酸合成在疟原虫肝期发育过程中起着关键作用

Falkard Brie, Kumar T R Santha, Hecht Leonie-Sophie, Matthews Krista A, Henrich Philipp P, Gulati Sonia, Lewis Rebecca E, Manary Micah J, Winzeler Elizabeth A, Sinnis Photini, Prigge Sean T, Heussler Volker, Deschermeier Christina, Fidock David

In vitro and in vivo activity of frenolicin B against Plasmodium falciparum and P berghei

弗雷诺林B对恶性疟原虫和伯氏疟原虫的体外和体内活性

Fitzgerald, Jay T; Henrich, Philipp P; O'Brien, Connor; Krause, Michael; Ekland, Eric H; Mattheis, Corinna; Sá, Juliana M; Fidock, David; Khosla, Chaitan