日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Biological Evaluation of Colibactin Derivatives

大肠杆菌素衍生物的合成及生物学评价

Airan, Yougant; Fedorova, Olga; Heer, Collin; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Bindra, Ranjit S; Herzon, Seth B

Targeted CRISPR knockout screening identifies known and novel chemogenomic interactions between DNA damaging agents and DNA repair genes

靶向 CRISPR 基因敲除筛选可识别 DNA 损伤剂与 DNA 修复基因之间已知的和新的化学基因组学相互作用

Heer, Collin D; Elia, James L; Menon, Vijay; Johnson, Spenser S; Arbelaez, Sofia R; Friedman, Sam; Lopez-Giraldez, Francesc; Sundaram, Ranjini K; Herzon, Seth B; Bindra, Ranjit S; Gueble, Susan E

Three-component assembly and structure-function relationships of (-)-gukulenin A

(-)-古库列宁A的三组分组装和结构-功能关系

Gupta, Vaani; Wang, Zechun; Combs, Joshua B; Wright, Timothy; Chen, Lei; Lin, Boxu; Holmes, Ryan; Qin, Bo; Oh, Joonseok; Crawford, Jason M; Herzon, Seth B

The Fanconi anemia pathway repairs colibactin-induced DNA interstrand cross-links

范可尼贫血通路修复大肠杆菌素诱导的DNA链间交联

Altshuller, Maria; He, Xu; MacKrell, Elliot J; Wernke, Kevin M; Airan, Yougant; Wong, Joel W H; Sellés-Baiget, Selene; Wang, Ting-Yu; Chou, Tsui-Fen; Duxin, Julien P; Balskus, Emily P; Herzon, Seth B; Semlow, Daniel R

Colibactin Exerts Androgen-dependent and -independent Effects on Prostate Cancer

大肠杆菌素对前列腺癌具有雄激素依赖性和非依赖性作用

Agrawal, Raag; Al-Hiyari, Sarah; Hugh-White, Rupert; Hromas, Robert; Patel, Yash; Williamson, Elizabeth A; Mootor, Mohammed F E; Gonzalez, Alfredo; Fu, Jianmin; Haas, Roni; Jordan, Madison; Wickes, Brian L; Mohammed, Ghouse; Tian, Mao; Doris, Molly J; Jobin, Christian; Wernke, Kevin M; Pan, Yu; Yamaguchi, Takafumi N; Herzon, Seth B; Boutros, Paul C; Liss, Michael A

A Stereoselective Oxidative Dimerization En Route to (-)-Lomaiviticin A

立体选择性氧化二聚反应合成(-)-洛马维替辛A

DiBello, Mikaela; Xu, Zhi; Palazzo, Alexandria M; Herzon, Seth B

Genome-scale CRISPR/Cas9 screening reveals the role of PSMD4 in colibactin-mediated cell cycle arrest.

基因组规模的 CRISPR/Cas9 筛选揭示了 PSMD4 在大肠杆菌素介导的细胞周期阻滞中的作用

Dougherty Michael W, Hoffmann Ryan M, Hernandez Maria C, Airan Yougant, Gharaibeh Raad Z, Herzon Seth B, Yang Ye, Jobin Christian

Mechanism of Action of KL-50, a Candidate Imidazotetrazine for the Treatment of Drug-Resistant Brain Cancers

KL-50(一种用于治疗耐药性脑癌的候选咪唑并四嗪类药物)的作用机制

Huseman, Eric D; Lo, Anna; Fedorova, Olga; Elia, James L; Gueble, Susan E; Lin, Kingson; Sundaram, Ranjini K; Oh, Joonseok; Liu, Jinchan; Menges, Fabian; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Batista, Victor S; Crawford, Jason M; Pyle, Anna M; Bindra, Ranjit S; Herzon, Seth B

Intramolecular Oxyalkylation of Unactivated Alkenes

未活化烯烃的分子内氧烷基化

Xu, Zhi; Airan, Yougant; Tomanik, Martin; Yang, Andrew T; Bhak, Natalie; Herzon, Seth B

Structure Elucidation of Secondary Metabolites: Current Frontiers and Lingering Pitfalls

次级代谢产物的结构解析:当前前沿进展与尚存挑战

DiBello, Mikaela; Healy, Alan R; Nikolayevskiy, Herman; Xu, Zhi; Herzon, Seth B