日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Light-aversion and cephalic allodynia in an intravenous CGRP model of migraine-like behaviour in male and female rats

在雄性和雌性大鼠的静脉注射 CGRP 偏头痛样行为模型中,光厌恶和头颅异常性疼痛

Andersen, Veronika K; Hansen, Bjarke S; Fungbrant, Emelie; Hestehave, Sara; Haanes, Kristian A; Nordahl, Karin M L

Analgesia through FKBP51 inhibition at disease onset confers lasting relief from sensory and emotional chronic pain symptoms.

在疾病发作时通过抑制 FKBP51 来达到镇痛效果,可以持久缓解感觉和情绪方面的慢性疼痛症状。

Hestehave Sara, Florea Roxana, Singleton Samuel, Fedorec Alex J H, Caxaria Sara, Morgan Oakley B, Kopp Katharina Tatjana, Brown Laurence A, Heymann Tim, Sikandar Shafaq, Hausch Felix, Peirson Stuart N, Géranton Sandrine M

Small molecule targeting Na V 1.7 via inhibition of CRMP2-Ubc9 interaction reduces pain-related outcomes in a rodent osteoarthritic model.

通过抑制 CRMP2-Ubc9 相互作用靶向 Na V 1.7 的小分子可减轻啮齿动物骨关节炎模型中的疼痛相关结果

Hestehave Sara, Allen Heather N, Gomez Kimberly, Duran Paz, Calderon-Rivera Aida, Loya-López Santiago, Rodríguez-Palma Erick J, Khanna Rajesh

Refining the adjuvant-induced rat model of monoarthritis by optimizing the induction volume and injection site

通过优化诱导体积和注射部位,改进佐剂诱导的大鼠单关节炎模型

Berke, Mie S; Hansen, Christian P; Kromann, Sofie; Colding-Jørgensen, Pernille; Kalliokoski, Otto; Jensen, Henrik E; Sørensen, Dorte Bratbo; Hau, Jann; Abelson, Klas S P; Hestehave, Sara

Quinoline-Based Neuropilin‑1 Antagonists Exhibit a Pure Antagonist Profile and Block Vascular Endothelial Growth Factor-Induced Pain

基于喹啉的神经纤毛蛋白-1拮抗剂表现出纯拮抗剂特性,并能阻断血管内皮生长因子诱导的疼痛。

Hestehave, Sara; Dragoni, Silvia; Fallon, Philip; Mota, Filipa; Calderon-Rivera, Aida; Gomez, Kimberly; Powell, Jonathan; Patsiarika, Anastasia; Reisinger, Tifelle; Crosby, Stuart; Chan, A W Edith; Steadman, David; Winfield, Natalie; Jarvis, Ashley; Martin, John; Zachary, Ian C; Frankel, Paul; Djordjevic, Snezana; Ruhrberg, Christiana; Khanna, Rajesh; Selwood, David L

C-H Functionalization-Enabled 11-Step Semisynthesis of (-)-Veragranine A and Characterization of Synthetic Analogs in Osteoarthritis-related Pain Treatment

CH 官能化实现的 11 步半合成 (-)-维拉格拉宁 A 及其合成类似物在骨关节炎相关疼痛治疗中的表征

Ma, Donghui; Duran, Paz; Al-Ahmad, Reem; Hestehave, Sara; Joa, Margarita; Alsbiei, Omar; Rodríguez-Palma, Erick J; Li, Yanrong; Wang, Shilin; Khanna, Rajesh; Dai, Mingji

C2230, a preferential use- and state-dependent CaV2.2 channel blocker, mitigates pain behaviors across multiple pain models.

C2230 是一种优先使用和状态依赖的 CaV2.2 通道阻滞剂,可减轻多种疼痛模型中的疼痛行为

Tang Cheng, Gomez Kimberly, Chen Yan, Allen Heather N, Hestehave Sara, Rodríguez-Palma Erick J, Loya-Lopez Santiago, Calderon-Rivera Aida, Duran Paz, Nelson Tyler S, Kanumuri Siva Rama Raju, Shah Bijal, Panigrahi Nihar R, Perez-Miller Samantha, Schackmuth Morgan K, Ruparel Shivani, Patwardhan Amol, Price Theodore J, Arora Paramjit S, Sharma Ravindra K, Sharma Abhisheak, Yu Jie, Korczeniewska Olga A, Khanna Rajesh

Reliability of sucrose preference testing following short or no food and water deprivation-a Systematic Review and Meta-Analysis of rat models of chronic unpredictable stress

短期或完全禁食禁水后蔗糖偏好测试的可靠性——慢性不可预测应激大鼠模型的系统评价和荟萃分析

Berrio, Jenny P; Hestehave, Sara; Kalliokoski, Otto

Uncoupling the CRMP2-Ca(V)2.2 Interaction Reduces Pain-Like Behavior in a Preclinical Joint-Pain Model.

解耦 CRMP2-Ca(V)2.2 相互作用可减少临床前关节疼痛模型中的疼痛样行为

Allen Heather N, Hestehave Sara, Duran Paz, Nelson Tyler S, Khanna Rajesh

Differences in multidimensional phenotype of 2 joint pain models link early weight-bearing deficit to late depressive-like behavior in male mice

两种关节疼痛模型的多维表型差异表明,雄性小鼠早期负重不足与后期抑郁样行为相关。

Hestehave, Sara; Florea, Roxana; Fedorec, Alexander J H; Jevic, Maria; Mercy, Lucile; Wright, Annia; Morgan, Oakley B; Brown, Laurence A; Peirson, Stuart N; Géranton, Sandrine M