C2230, a preferential use- and state-dependent CaV2.2 channel blocker, mitigates pain behaviors across multiple pain models.
C2230 是一种优先使用和状态依赖的 CaV2.2 通道阻滞剂,可减轻多种疼痛模型中的疼痛行为
期刊:Journal of Clinical Investigation
影响因子:13.6
doi:10.1172/JCI177429
Tang Cheng, Gomez Kimberly, Chen Yan, Allen Heather N, Hestehave Sara, RodrÃguez-Palma Erick J, Loya-Lopez Santiago, Calderon-Rivera Aida, Duran Paz, Nelson Tyler S, Kanumuri Siva Rama Raju, Shah Bijal, Panigrahi Nihar R, Perez-Miller Samantha, Schackmuth Morgan K, Ruparel Shivani, Patwardhan Amol, Price Theodore J, Arora Paramjit S, Sharma Ravindra K, Sharma Abhisheak, Yu Jie, Korczeniewska Olga A, Khanna Rajesh