日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

Exploiting the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists

利用 2-(1,3,4,9-四氢吡喃并[3,4-b]吲哚-1-基)乙酸骨架生成 COXTRANs:一类新型双重环氧合酶抑制剂-血栓素受体拮抗剂

Blua, Federica; Boccato, Francesca; Buccellati, Carola; Risè, Patrizia; Barbieri, Silvia; Castiglioni, Laura; Balzulat, Annika; Rolando, Barbara; Marini, Elisabetta; Balestra, Marta; Introvigne, Maria Luisa; Giorgis, Marta; Sironi, Luigi; Tacconelli, Stefania; Hiesinger, Kerstin; Patrignani, Paola; Schmidtko, Achim; Steinhilber, Dieter; Proschak, Ewgenij; Sala, Angelo; Rovati, G Enrico; Bertinaria, Massimo

Structure-Based Design of PROTACS for the Degradation of Soluble Epoxide Hydrolase.

基于结构的PROTACS设计用于降解可溶性环氧化物水解酶

Schönfeld Julia, Brunst Steffen, Ciomirtan Ludmila, Willmer Lena, Chromik Michel A, Kumar Adarsh, Froemel Timo, Liebisch Nick, Hackspacher Arne, Ehrler Johanna H M, Wintermeier Lukas, Hesse Christina, Fiedler Jan, Heering Jan, Freitag Hinrich, Zardo Patrick, Fieguth Hans-Gerd, Brüggerhoff Astrid, Jakob Josefine, Häupl Björn, Weizel Lilia, Kaiser Astrid, Schubert-Zsilavecz Manfred, Oellerich Thomas, Fleming Ingrid, Schebb Nils H, Fürst Robert, Kannt Aimo, Knapp Stefan, Proschak Ewgenij, Hiesinger Kerstin

Designing a Small Fluorescent Inhibitor to Investigate Soluble Epoxide Hydrolase Engagement in Living Cells

设计一种小型荧光抑制剂来研究活细胞中可溶性环氧化物水解酶的活性

Brunst, Steffen; Schönfeld, Julia; Breunig, Peter; Burgers, Luisa D; DeMeglio, Murphy; Ehrler, Johanna H M; Lillich, Felix F; Weizel, Lilia; Hefendehl, Jasmin K; Fürst, Robert; Proschak, Ewgenij; Hiesinger, Kerstin

Systematic Assessment of Fragment Identification for Multitarget Drug Design

多靶点药物设计中片段识别的系统性评估

Brunst, Steffen; Kramer, Jan S; Kilu, Whitney; Heering, Jan; Pollinger, Julius; Hiesinger, Kerstin; George, Sven; Steinhilber, Dieter; Merk, Daniel; Proschak, Ewgenij